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958226-81-8

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "958226-81-8" in MCE Product Catalog:

Cat. No.: HY-158618
CAS No.: 958226-81-8
Target:  

Aurora Kinase Apoptosis

Research Areas:  

Cancer

Aurora kinase inhibitor-14 (Compound 79) is an orally active and highly selective inhibitor of Aurora kinases with IC50 values of 0.5 nM and 1.2 nM for Aurora A and Aurora B, respectively. Aurora kinase inhibitor-14 binds to the ATP-binding site of Aurora kinases to block chromosome segregation during mitosis and induce apoptosis in tumor cells. Aurora kinase inhibitor-14 is promising for research of various solid tumors and hematological malignancies, such as non-small cell lung cancer, breast cancer, and acute myeloid leukemia .
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