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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
2 Results for "
AR antagonist 15
" in MedChemExpress (MCE) Product Catalog:
Products (2)
2 Results for "AR antagonist 15" in MCE Product Catalog:
Cat. No.: HY-174391
CAS No.: 1790308-86-9
Target:
Research Areas:
AR antagonist 15 is an orally active androgen receptor (AR) antagonist with the IC50 of 97 nM for ART787A. AR antagonist 15 disrupts AR nuclear translocation, hinders AR homodimerization, and suppresses transcription of AR-regulated genes by competitive binding to the ligand binding pocket. AR antagonist 15 can significantly lower the prostate-specific antigen (PSA) level. AR antagonist 15 induces apoptosis by reducing the expression of apoptosis pathway related proteins. AR antagonist 15 can be used for the research of prostate cancer.
Cat. No.: HY-184957
CAS No.: 3033660-79-3
Research Areas:
Androgen receptor antagonist 15 is an Androgen receptor (AR) antagonist. Androgen receptor antagonist 15 serves as a Ligand for Target Protein for PROTAC for PROTAC AR degraders, such as ARD-61 (HY-139659). Androgen receptor antagonist 15 is applicable to the research of prostate cancer .
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Protocols
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