3 Results for "

Androgen receptor-IN-5

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Androgen receptor-IN-5" in MCE Product Catalog:

Cat. No.: HY-153276
CAS No.: 1391944-16-3
Target:  

Androgen Receptor

Research Areas:  

Cancer

Androgen receptor-IN-5 is an androgen receptor inhibitor with potent anticancer effects. Androgen receptor-IN-5 also inhibits the production of IL-17A, IL- 17F and INF-γ (WO2023281097A1,Example 1/1) .
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Cat. No.: HY-162764
CAS No.: 2902679-11-0
Target:  

Androgen Receptor

Research Areas:  

Cancer

Androgen receptor degrader-5 is an androgen receptor (AR) degrader. Androgen receptor degrader-5 induces proteasome-dependent degradation of androgen receptor protein and inhibits the transcriptional activity of wild-type AR and AR F876L. Androgen receptor degrader-5 exhibits anticancer activity against prostate cancer. Androgen receptor degrader-5 can be used in the research of prostate cancer .
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Cat. No.: HY-146494
CAS No.: 2586195-28-8
Target:  

Androgen Receptor

Research Areas:  

Cancer

Androgen receptor antagonist 5 (compound 42f) is a potent androgen receptor (AR) antagonist with an IC50 value of 6.17 μM. Androgen receptor antagonist 5 can effectively impair AR nuclear translocation, reducing the levels of nuclear AR, and disrupts AR-mediated gene regulation. Androgen receptor antagonist 5 has antiproliferative activity against LNCaP and exhibits antitumor activity in LNCaP xenograft tumor mice model. Androgen receptor antagonist 5 can be used for researching prostate cancer .
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