1 Result for "

Glucocorticoid receptor modulator5

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Glucocorticoid receptor modulator5" in MCE Product Catalog:

Cat. No.: HY-181014
Glucocorticoid receptor modulator 5 (Compound D8) is a selective, orally active Glucocorticoid receptor modulator. Glucocorticoid receptor modulator 5 shows extremely high transrepression activity (TRNF-κB IC50 = 0.0009 μM, TRAP-1 IC50 = 0.0005 μM). Glucocorticoid receptor modulator 5 exerts its anti-inflammatory activity by interacting directly with the Glucocorticoid receptor signaling pathway. Glucocorticoid receptor modulator 5 significantly alleviates dermatitis and autoimmune hepatitis .
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