Glucocorticoid receptor modulator 5
Glucocorticoid receptor modulator 5 (Compound D8) is a selective, orally active Glucocorticoid receptor modulator. Glucocorticoid receptor modulator 5 shows extremely high transrepression activity (TRNF-κB IC50 = 0.0009 μM, TRAP-1 IC50 = 0.0005 μM). Glucocorticoid receptor modulator 5 exerts its anti-inflammatory activity by interacting directly with the Glucocorticoid receptor signaling pathway. Glucocorticoid receptor modulator 5 significantly alleviates dermatitis and autoimmune hepatitis.
For research use only. We do not sell to patients.
- Formula: C24H23ClN2O4S
- Molecular Weight:470.97
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Biological Activity
Chemical Information
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Molecular Weight 470.97
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Formula C24H23ClN2O4S
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SMILES
O=S(NC1=CC=C2N(C(CCC2=C1)=O)CC3=CC=CC=C3)(C4=CC(Cl)=C(C=C4OC)C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Glucocorticoid receptor modulator 5 Related Classifications
HY-181014 Related Classifications
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