5 Results for "

Human vas deferens

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "Human vas deferens" in MCE Product Catalog:

Cat. No.: HY-118335
CAS No.: 107021-36-3
Purity:  96.20%
Synonyms: SZL 49
Target:  

Adrenergic Receptor

Research Areas:  

Cardiovascular Disease

Prazobind (SZL 49), a prazosin analog, is an irreversible α1-adrenoceptor antagonist. Prazobind competes for alpha 1-adrenoceptor binding sites with a similar potency (IC50 of 1 nM) in tissues enriched in both the alpha 1A (hippocampus) and alpha 1B (liver) subtypes. Prazobind partially inhibits the contractions of circular muscles, longitudinal muscles and smooth muscles of the spleen. Prazobind can be used for the study of blood pressure .
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Cat. No.: HY-P3679
CAS No.: 131448-51-6
Research Areas:  

Neurological Disease

Neuropeptide Y (1-24) (human) is a neuropeptide with potencies in inhibiting the electricity stimulated twitch response of rat vas deferens. Neuropeptide Y (1-24) (human) stimulates N-methyl-D-aspartate (NMDA)-induced neuronal activation in the rat CA3 region of the dorsal hippocampus in vivo .
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Cat. No.: HY-P2601A
Target:  

CGRP Receptor

Research Areas:  

Others

Tyr-α-CGRP (human) TFA is an N-terminally extended human α-CGRP analog. Tyr-α-CGRP (human) TFA can bind to membrane preparations from rat brain and spleen with IC50 values of 0.2 nM and 0.5 nM, respectively, and induce positive chronotropic and inotropic effects in isolated guinea pig right and left atria with EC50 values of 282 nM and 74 nM, respectively. Tyr-α-CGRP (human) TFA also inhibits contractile responses in rat vas deferens with an EC50 value of 1.9 nM .
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Cat. No.: HY-N9554
CAS No.: 150881-27-9
WIN-64821 is a secondary metabolite produced by Aspergillus species, and acts as a Neurokinin Receptor antagonist. The Ki values of WIN-64821 for NK1, NK2 and NK3 receptors are 0.24 (human astrocytoma cells), 0.26 (rat duodenum) and 15.2 (guinea pig forebrain) μM, respectively. WIN-64821 inhibits apamin-induced contraction of rat vas deferens, blocks substance P-induced contraction of guinea pig ileum and Ca 2+ efflux in human astrocytoma cells. WIN-64821 is applicable to analgesic and anti-inflammatory research .
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Cat. No.: HY-W745352
CAS No.: 65-15-6
Target:  

Adrenergic Receptor

Azapetine hydrochloride is a selective α1-adrenergic receptor inhibitor with an IC50 of 205 nM. Azapetine hydrochloride inhibits Epinephrine (HY-B0447)-induced platelet aggregation, slightly enhances the contractile response of isolated rat vas deferens, and blocks α1 and α2 adrenergic receptor-mediated vasoconstriction .
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