13 Results for "

indolocarbazole

" in MedChemExpress (MCE) Product Catalog:
Products (13)

13 Results for "indolocarbazole" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-149266
CAS No.: 2226941-26-8
Purity:  99.80%
Target:  

ROCK

Research Areas:  

Cancer

THK01 is a potent ROCK2 inhibitor with IC50 values of 5.7 and 923 nM for ROCK2 and ROCK1, respectively. THK01 inhibits breast cancer metastasis through the ROCK2-STAT3 signaling pathway. THK01 can be used in research of breast cancer .
loading...
    loading...
Cat. No.: HY-P1726
CAS No.: 1416983-77-1
MSG606 is a selective melanocortin 1 receptor (MC1R) antagonist. MSG606 can abolish the neuroprotective effects of BMS-470539 (HY-15616) (MC1R agonist). MSG606 can inhibit cancer cell proliferation and transition from the G1 to the S phase. MSG606 can delay pain hypersensitivity and reduce cholesterol levels. MSG606 can be used for the researches of cancer, inflammation, neurological and metabolic disease, such as breast cancer and subarachnoid hemorrhage (SAH) .
loading...
    loading...
Cat. No.: HY-N16039
CAS No.: 126221-76-9
TAN-1030A is an indolocarbazole alkaloid with macrophage-activating properties. TAN-1030A induces spreading of a murine macrophage cell line, Mm 1, and augmentes the phagocytic activity, Fc gamma receptor expression and β-glucuronidase activity of murine macrophage cell lines, Mm 1 and J774A.1. TAN-1030A can activate macrophage functions in mice .
loading...
    loading...
Cat. No.: HY-P0077
CAS No.: 1190083-57-8
Target:  

Oxytocin Receptor

Research Areas:  

Endocrinology

Merotocin is a selective, short-acting peptidic oxytocin receptor agonist. Merotocin can be used to support lactation .
loading...
    loading...
Cat. No.: HY-P1726A
MSG606 TFA is a selective melanocortin 1 receptor (MC1R) antagonist. MSG606 TFA can abolish the neuroprotective effects of BMS-470539 (HY-15616) (MC1R agonist). MSG606 TFA can inhibit cancer cell proliferation and transition from the G1 to the S phase. MSG606 TFA can delay pain hypersensitivity and reduce cholesterol levels. MSG606 TFA can be used for the researches of cancer, inflammation, neurological and metabolic disease, such as breast cancer and subarachnoid hemorrhage (SAH) .
loading...
    loading...
Cat. No.: HY-P0041A
Target:  

Vasopressin Receptor

Research Areas:  

Neurological Disease

F992 TFA is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue .
loading...
    loading...
Cat. No.: HY-N6734
CAS No.: 99570-78-2
K-252b, an indolocarbazole isolated from the actinomycete Nocardiopsis, is a PKC inhibitor. K-252b can be used to inhibit extracellular kinases of cells in culture because it can’t pass through cell membrane freely .
loading...
    loading...
Cat. No.: HY-130748
CAS No.: 105114-22-5
Research Areas:  

Infection

K-252d is an indolocarbazole alkaloid found in Nocardiopsis. It is a PKC inhibitor that inhibits PKC isolated from rat brain (IC50=350 nM). It also inhibits calcium- and calmodulin-dependent phosphodiesterase isolated from bovine heart (IC50=46.2 μM).
loading...
    loading...
Cat. No.: HY-P2331
CAS No.: 59165-34-3
Synonyms: Antibiotic A 3802-IV-3; Gardimycin
Target:  

Antibiotic

Research Areas:  

Infection

Actagardin is a tetracyclic lantibiotic produced by several species of Actinoplanes. It is composed of macrocyclic rings formed by thioether bridges. Actagardin preferably targets Gram-positive bacteria, inhibiting the synthesis of peptidoglycan.
loading...
    loading...
Cat. No.: HY-P10014
CAS No.: 153507-46-1
Target:  

Peptides

Research Areas:  

Cardiovascular Disease

Bibapcitide, a 26 amino acid, inhibits thrombosis .
loading...
    loading...
Cat. No.: HY-P0041
CAS No.: 162277-99-8
Target:  

Vasopressin Receptor

Research Areas:  

Neurological Disease

F992 is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue .
loading...
    loading...
Cat. No.: HY-P4948
CAS No.: 1926163-49-6
Research Areas:  

Others

Coumarin-phalloidin is a kind of phalloidin labeled with Coumarin (HY-N0709). Coumarin-phalloidin is a new type of actin probe that can be used for triple immunofluorescence microscopic observation of the cell skeleton .
loading...
    loading...
Cat. No.: HY-P11823
Target:  

Fluorescent Dye

Research Areas:  

Inflammation/Immunology Cancer

FAPα/DPP4 fluorogenic substrate-1 is a fluorogenic macrocyclic peptide substrate that can be cleaved by FAPα and DPP4. FAPα/DPP4 fluorogenic substrate-1 can be used in the research of cancer and type 2 diabetes .
loading...
    loading...
  • 1