21 Results for "

opioid derivative

" in MedChemExpress (MCE) Product Catalog:
Products (21)

21 Results for "opioid derivative" in MCE Product Catalog:

Cat. No.: HY-W013154
CAS No.: 136030-33-6
Research Areas:  

Others

Fmoc-Tic-OH, an Fmoc-protected derivative of Tic, is a solid-phase peptide synthesis monomer. Fmoc-Tic-OH protects the amino group of Tic via a base-labile Fmoc group, allowing conformationally constrained Tic residues to be stepwise coupled to peptide chains, and the Fmoc protecting group can be removed under piperidine conditions. Fmoc-Tic-OH can be used for peptide synthesis and opioid receptor ligand research .
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Cat. No.: HY-W048697
CAS No.: 201532-01-6
Research Areas:  

Others

Fmoc-D-Pen(Trt)-OH is an amino acid derivative with an Fmoc protecting group, which can be used to synthesize analogs of cyclic lanthionine enkephalin, a δ-opioid receptor selective ligand .
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Cat. No.: HY-136208
CAS No.: 892039-23-5
Purity:  99.44%
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

TAN-452 is an orally active, selective peripherally acting δ-opioid receptor (DOR) antagonist with a Ki of 0.47 nM and a Kb of 0.21 nM. TAN-452 is an antagonist for μ-opioid receptor (MOR; Ki=36.56 nM and Kb=9.43 nM) and κ-opioid receptor (KOR; Ki=5.31 nM and Kb=7.18 nM). TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control .
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Cat. No.: HY-W000665
CAS No.: 123715-02-6
Synonyms: Dmt
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

2,6-Dimethyl-L-tyrosine (Dmt) is a tyrosine derivative that enhances receptor affinity, functional bioactivity and in vivo analgesia of opioid peptides .
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Cat. No.: HY-D1387
CAS No.: 2080300-52-1
Naloxone fluorescein acetate is the fluorescent-derivative of Naloxone. Naloxone is an opioid antagonist. Naloxone is the antidote for reversing the effects of an opioid overdose .
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Cat. No.: HY-P3632
CAS No.: 75921-88-9
Synonyms: DADAD
Target:  

Opioid Receptor

[DAla2, DArg6] Dynorphin A, (1-13) (porcine) (DADAD) is an opioid peptide (dynorphinl-13, DYN) derivative found in porcine pituitary extracts. DYN is highly potent at the peripheral opioid receptors GPI and MVD, but is readily and rapidly degraded in vivo. [DAla2, DArg6] Dynorphin A, (1-13) (porcine) has some resistance to enzymatic cleavage and prevents peptide cleavage by enzymes .
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Cat. No.: HY-172560
Target:  

Drug Metabolite

6β-Oxycodol N-oxide is an opioid derivative and a metabolite of Oxycodone, which can be detected in urine .
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Cat. No.: HY-128624
CAS No.: 2361560-81-6
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

DS39201083, a Conolidine derivative, is a potent and orally active analgesic agent. DS39201083 shows no agonist activity at the mu opioid receptor. DS39201083 can be used for the study of neurological diseases .
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Cat. No.: HY-113683
CAS No.: 1018988-00-5
Synonyms: AZD7268
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

AZ 12488024 (AZD7268) is a SNC80 (HY-101202) derivative and a δ-opioid receptor agonist. AZ 12488024 is available for research into major depressive disorder .
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Cat. No.: HY-P3625
CAS No.: 161874-98-2
Dynorphin (2-17), amide (porcine) is a dynorphin derivative with some analgesic effects. Dynorphin is a class of opioid peptides produced by the precursor protein dynorphinogen and is involved in pain, addiction and mood regulation .
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Cat. No.: HY-162570
CAS No.: 15686-68-7
Target:  

Opioid Receptor

Research Areas:  

Others

Volazocine is an opioid benzomorphane derivative with potential analgesic activity .
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Cat. No.: HY-106873A
CAS No.: 22443-55-6
Purity:  99.59%
Target:  

Drug Derivative

Research Areas:  

Others

Nepinalone hydrochloride, an alchilaminate derivative of β-tetralone and an orally active cough suppressant, possesses a non-opioid antitussive activity .
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Cat. No.: HY-106873
CAS No.: 22443-11-4
Target:  

Drug Derivative

Research Areas:  

Others

Nepinalone, an alchilaminate derivative of β-tetralone and an orally active cough suppressant, possesses a non-opioid antitussive activity .
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Cat. No.: HY-100963
CAS No.: 112465-94-8
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

U-54494A is a benzamide derivative related to κ-opioid receptor agonists, U-54494A has an anticonvulsant activity .
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Cat. No.: HY-142918
CAS No.: 2667632-83-7
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

μ opioid receptor agonist 1 (Compound H-1a)is an optically pure oxaspiro ring substituted pyrrolopyrazole derivative, acts as a MOR receptor agonist and can be used for the research of pain and pain related diseases .
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Cat. No.: HY-142919
CAS No.: 2671755-38-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

μ opioid receptor agonist 2 (Compound H-3)is an optically pure oxaspiro ring substituted pyrrolopyrazole derivative, acts as a MOR receptor agonist and can be used for the research of pain and pain related diseases .
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Cat. No.: HY-P3647
CAS No.: 94596-26-6
Research Areas:  

Neurological Disease

[DPro10] Dynorphin A (1-11), porcine, a N-Alkylated derivative, is a potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine has analgesic property .
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Cat. No.: HY-P3647A
Research Areas:  

Neurological Disease

[DPro10] Dynorphin A (1-11), porcine hydrochloride, a N-Alkylated derivative, is a potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine hydrochloride has analgesic property .
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Cat. No.: HY-P10555
CAS No.: 90549-86-3
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

(D-Arg2, Sar 4)-Dermorphin (1-4) is a tetrapeptide derivative of the peptide Dermorphin (HY-P0244) found in amphibian skin. (D-Arg2, Sar 4)-Dermorphin (1-4) has significant analgesic effects by binding to the μ-opioid receptor (MOR) in the body. (D-Arg2, Sar 4)-Dermorphin (1-4) can be used in the development of analgesic drugs .
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Cat. No.: HY-179365
CAS No.: 63463-07-0
Synonyms: β-NTA dihydrochloride
Target:  

Drug Intermediate

Research Areas:  

Others

β-Naltrexamine (β-NTA) dihydrochloride is a key synthetic intermediate used in the preparation of irreversible ligands for opioid receptors .
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