AKR1C2/3-IN-1
AKR1C2/3-IN-1 (compound 3a) is a potent AKR1C2 and AKR1C3 inhibitor with IC50 values of 90, 50 nM, respectively. AKR1C2/3-IN-1 can be used as a radiation sensitizer and as a potentiator of chemotherapy cytotoxicity.
For research use only. We do not sell to patients.
- CAS No.: 3107747-45-2
- Formula: C14H15NO4
- Molecular Weight:261.27
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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AKR1C3 50 nM (IC50) |
AKR1C2 90 nM (IC50) |
Chemical Information
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CAS No. 3107747-45-2
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Molecular Weight 261.27
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Formula C14H15NO4
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SMILES
O=C(C(C1=O)=CC2=C(O1)C=C(O)C=C2)N(CC)CC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)