1143024-28-5
Chemical Structure
GPR81 agonist 2
- CAS No.: 1143024-28-5
- Formula:C26H27ClN6O5S2
- Molecular Weight:603.11
InChIKey: ZVDDZDATCIKPCU-UHFFFAOYSA-N
SMILES: O=C(NC1=NC2=C(S1)C=C(S(=O)(C3CCN(CC3)C)=O)C=C2)NC(C4=C(Cl)C=C(OCC)C(N5N=CC=C5)=C4)=O
Biological Activity: GPR81 agonist 2 is a GPR81 agonist with an EC50 of 0.023 μM for the human receptor. GPR81 agonist 2 activates the lactate-sensing receptor GPR81, inhibits forskolin-stimulated cAMP production and GTP binding of Gi protein. GPR81 agonist 2 can be used for research on type 2 diabetes[1].
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GPR81 agonist 2 | GPR81 agonist 2 is a GPR81 agonist with an EC50 of 0.023 μM for the human receptor. GPR81 agonist 2 activates the lactate-sensing receptor GPR81, inhibits forskolin-stimulated cAMP production and GTP binding of Gi protein. GPR81 agonist 2 can be used for research on type 2 diabetes. | |||||||||||||||||||||
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