3032750-17-4
Chemical Structure
DS69910557
- CAS No.: 3032750-17-4
- Formula:C32H33Cl2FN4O3
- Molecular Weight:611.53
IUPAC Name: (1r,4r)-4-(((1-(4-(2,9-dichloro-5,5-dimethyl-6-oxo-5,6-dihydro-7H-benzo[b]pyrido[3,2-d]azepin-7-yl)phenyl)-3-fluoroazetidin-3-yl)methyl)amino)cyclohexane-1-carboxylic acid
InChIKey: JAOGFYSXDYNYSX-XYWHTSSQSA-N
SMILES: ClC(C=N1)=CC(C2=C(C=C(Cl)C=C2)N3C4=CC=C(N5CC(F)(CN[C@@H]6CC[C@@H](C(O)=O)CC6)C5)C=C4)=C1C(C)(C)C3=O
Biological Activity: DS69910557 is a potent, selective and orally activehuman parathyroid hormone receptor 1 (hPTHR1) antagonist. DS69910557 has antagonistic activity for PTHR1 with an IC50 value of 0.08 μM. DS69910557 can be used for the research of hyperparathyroidism, hypercalcemia of malignancy and osteoporosis[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DS69910557 | 98.86% | DS69910557 is a potent, selective and orally activehuman parathyroid hormone receptor 1 (hPTHR1) antagonist. DS69910557 has antagonistic activity for PTHR1 with an IC50 value of 0.08 μM. DS69910557 can be used for the research of hyperparathyroidism, hypercalcemia of malignancy and osteoporosis. | ||||||||||||||||||||
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Keywords
