371962-01-5
371962-01-5
Chemical Structure
ZAPA sulfate
- CAS No.: 371962-01-5
- Formula:C4H8N2O6S2
- Molecular Weight:244.25
IUPAC Name: (Z)-3-(carbamimidoylthio)acrylic acid compound with sulfuric acid (1:1)
InChIKey: UWVNHPNVOMFDHW-ODZAUARKSA-N
SMILES: O=C(O)/C=C\SC(N)=N.O=S(O)(O)=O
Biological Activity: ZAPA sulfate is an agonist at low affinity GABAA-receptors. ZAPA sulfate induces membrane hyperpolarization of the Ascaris muscle cell with an EC50 of 10.3 μM[1][2].
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ZAPA sulfate | 99.25% | ZAPA sulfate is an agonist at low affinity GABAA-receptors. ZAPA sulfate induces membrane hyperpolarization of the Ascaris muscle cell with an EC50 of 10.3 μM. | ||||||||||||||||||||
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ZAPA sulfate (Standard) | ≥98% | ZAPA (sulfate) (Standard) is the analytical standard of ZAPA (sulfate) (HY-100799). This product is intended for research and analytical applications. ZAPA sulfate is an agonist at low affinity GABAA-receptors. ZAPA sulfate induces membrane hyperpolarization of the Ascaris muscle cell with an EC50 of 10.3 μM. | ||||||||||||||||||||
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References
- [1]. Yokogawa T, et al. Analysis of GABAA‐and GABAB‐receptor mediated effects on intracellular Ca2+ in DRG hybrid neurones. British journal of pharmacology, 2001, 134(1): 98-107.
- [2]. Holden-Dye L, et al. ZAPA, (Z)-3-[(aminoiminomethyl)thio]-2-propenoic acid hydrochloride, a potent agonist at GABA-receptors on the Ascaris muscle cell. Br J Pharmacol. 1988 Sep;95(1):3-5. [Content Brief]
Keywords
