ZAPA sulfate

Cat. No.: HY-100799 Purity: 99.25%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

ZAPA sulfate is an agonist at low affinity GABA_A-receptors. ZAPA sulfate induces membrane hyperpolarization of the Ascaris muscle cell with an EC₅₀ of 10.3 μM.

For research use only. We do not sell to patients.

ZAPA sulfate Chemical Structure

CAS No. : 371962-01-5

Size	Price	Stock	Quantity
5 mg	USD 95	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 150	In-stock	Estimated Time of Arrival: December 31
25 mg	USD 320	In-stock	Estimated Time of Arrival: December 31
50 mg	USD 530	In-stock	Estimated Time of Arrival: December 31
100 mg	USD 890	In-stock	Estimated Time of Arrival: December 31
200 mg		Get quote
500 mg		Get quote

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Description

ZAPA sulfate is an agonist at low affinity GABA_A-receptors. ZAPA sulfate induces membrane hyperpolarization of the Ascaris muscle cell with an EC₅₀ of 10.3 μM^[1]^[2].

In Vitro

Local applications of ZAPA (100 μM) sulfate transiently increases [Ca²⁺]_i, similar to the GABA-evoked responses^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

244.25

Formula

C₄H₈N₂O₆S₂

CAS No.

371962-01-5

Appearance

Solid

Color

White to off-white

SMILES

O=C(O)/C=C\SC(N)=N.O=S(O)(O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : 31.25 mg/mL (127.94 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

H₂O : 1.64 mg/mL (6.71 mM; ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	4.0942 mL	20.4708 mL	40.9417 mL
5 mM	0.8188 mL	4.0942 mL	8.1883 mL
10 mM	0.4094 mL	2.0471 mL	4.0942 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.25%

Select Batch:

Data Sheet (273 KB) SDS (251 KB)

COA (249 KB) HNMR (227 KB) LCMS (306 KB)

Handling Instructions (2659 KB)

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

H₂O / DMSO	1 mM	4.0942 mL	20.4708 mL	40.9417 mL	102.3541 mL
H₂O / DMSO	5 mM	0.8188 mL	4.0942 mL	8.1883 mL	20.4708 mL
DMSO	10 mM	0.4094 mL	2.0471 mL	4.0942 mL	10.2354 mL
	15 mM	0.2729 mL	1.3647 mL	2.7294 mL	6.8236 mL
	20 mM	0.2047 mL	1.0235 mL	2.0471 mL	5.1177 mL
	25 mM	0.1638 mL	0.8188 mL	1.6377 mL	4.0942 mL
	30 mM	0.1365 mL	0.6824 mL	1.3647 mL	3.4118 mL
	40 mM	0.1024 mL	0.5118 mL	1.0235 mL	2.5589 mL
	50 mM	0.0819 mL	0.4094 mL	0.8188 mL	2.0471 mL
	60 mM	0.0682 mL	0.3412 mL	0.6824 mL	1.7059 mL
	80 mM	0.0512 mL	0.2559 mL	0.5118 mL	1.2794 mL
	100 mM	0.0409 mL	0.2047 mL	0.4094 mL	1.0235 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ZAPA371962-01-5Inhibitorinhibitorinhibit

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