PARP1-IN-47
PARP1-IN-47 (Compound 35) is a highly selective PARP1 inhibitor (IC50 <100 nM). PARP1-IN-47 blocks poly(ADP-ribosyl)ation and disrupts DNA damage repair pathways to induce tumor cell apoptosis. PARP1-IN-47 is promising for research of solid tumors and hematological malignancies.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 3053592-61-0
- Fòrmula: C21H24F3N7O2
- Peso molecular:463.46
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
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PARP1 <100 nM (IC50) |
Chemical Information
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No. CAS 3053592-61-0
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Peso molecular 463.46
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Fòrmula C21H24F3N7O2
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SMILES
O=C(N1)C(CC)=CN2C1=CC(CN3CCN(CC3)C4=C(C(F)(F)F)N=C(C(NC)=O)C=C4)=N2
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)