PARP Inhibitors

PARP

PARP1

PARP2

PARP3

PARP4

TNKS1/PARP5A

TNKS2/PARP5B

PARP7

PARP10

PARP14

PARP15

PARP12

PARP16

PARP Inhibitors, Activators, Inducers, Degraders & Ligands

Product Name	PARP	PARP1	PARP2	PARP3	PARP4	TNKS1/PARP5A	TNKS2/PARP5B	PARP7	PARP10	PARP14	PARP15	PARP12	PARP16	Purity
Olaparib		PARP-1, IC₅₀: 5 nM	PARP-2, IC₅₀: 1 nM			tankyrase-1, IC₅₀: 1.5 μM								99.98%
XAV-939		ARTD1, IC₅₀: 5500 nM	ARTD2, IC₅₀: 479 nM			TNKS1, IC₅₀: 5 nM	TNKS2, IC₅₀: 2 nM							99.91%
Talazoparib		PARP1, Ki: 1.2 nM	PARP2, Ki: 0.87 nM											99.89%
Niraparib		PARP-1, IC₅₀: 3.8 nM	PARP-2, IC₅₀: 2.1 nM	PARP-3, IC₅₀: 1300 nM	V-PARP, IC₅₀: 330 nM	TANK-1, IC₅₀: 570 nM								99.96%
PARP1-IN-56		PARP1												99.03%
Saruparib		PARP1, IC₅₀: 3 nM	PARP2, IC₅₀: 1400 nM											99.76%
Rucaparib		PARP-1, Ki: 1.4 nM												99.96%
Veliparib		PARP-1, Ki: 5.2 nM	PARP-2, Ki: 2.9 nM											99.77%
PJ34	PARP, IC₅₀: 110 nM	PARP-1, IC₅₀: 110 nM	PARP-2, IC₅₀: 86 nM											99.66%
RBN-2397								PARP-7, IC₅₀: 3 nM PARP-7, Kd: 1 nM						99.82%
IRF1-IN-1		PARP-1												99.72%
Fluzoparib		PARP-1, IC₅₀: 1.46±0.72 nM												99.96%
KSQ-4279		PARP1												99.96%
Pamiparib	PARP													99.96%
SK-575		PARP1, IC₅₀: 2.30 nM												99.86%
3-Aminobenzamide	PARP, IC₅₀: 50 nM													99.97%
Dehydrocorydaline	PARP													99.77%
RBN012759					PARP4, IC₅₀: 10 μM			PARP7, IC₅₀: 4 μM	PARP10, IC₅₀: 1 μM	PARP14, IC₅₀: <3 nM				99.33%
Niraparib hydrochloride		PARP-1, IC₅₀: 3.8 nM	PARP-2, IC₅₀: 2.1 nM	PARP-3, IC₅₀: 1300 nM	V-PARP, IC₅₀: 330 nM	TANK-1, IC₅₀: 570 nM								99.41%
WIKI4							TNKS2, IC₅₀: 26 nM							99.93%
Rucaparib phosphate		PARP-1, Ki: 1.4 nM												99.76%
NVP-TNKS656			PARP2, IC₅₀: 32 μM				TNKS2, IC₅₀: 6 nM							99.66%
Niraparib tosylate		PARP-1, IC₅₀: 3.8 nM	PARP-2, IC₅₀: 2.1 nM	PARP-3, IC₅₀: 1300 nM	V-PARP, IC₅₀: 330 nM	TANK-1, IC₅₀: 570 nM								99.99%
Peiminine		PARP-1												99.89%
Paris saponin VII		PARP-1												99.84%
IRF1-IN-2		PARP-1												99.83%
BGP-15	PARP, IC₅₀: 120 μM													99.57%
Triclabendazole	PARP													99.36%
G007-LK						TNKS1, IC₅₀: 46 nM	TNKS2, IC₅₀: 25 nM							99.24%
AG14361		PARP-1, Ki: 0.5 nM												99.42%
OUL232		PARP1, IC₅₀: 15 μM	PARP2, IC₅₀: 10 μM	PARP3, IC₅₀: 50 μM	PARP4, IC₅₀: 11 μM	TNKS1, IC₅₀: 5.4 μM	TNKS2, IC₅₀: 10 μM	PARP7, IC₅₀: 83 nM	PARP10, IC₅₀: 7.8 nM	PARP14, IC₅₀: 300 nM	PARP15, IC₅₀: 56 nM			99.86%
Stenoparib		PARP1, IC₅₀: 2 nM	PARP2, IC₅₀: 1 nM			TNKS1, IC₅₀: 50 nM	TNKS2, IC₅₀: 50 nM							98.0%
OUL35									ARTD10/PARP10, IC₅₀: 329 nM					99.80%
UPF 1069		PARP-1, IC₅₀: 8 μM	PARP-2, IC₅₀: 0.3 μM											99.02%
Rucaparib monocamsylate		PARP-1, Ki: 1.4 nM												99.91%
RBN-3143		PARP1, IC₅₀: >100000 nM	PARP2, IC₅₀: >100000 nM	PARP3, IC₅₀: >100000 nM	PARP4, IC₅₀: 42700 nM				PARP10, IC₅₀: 1600 nM	PARP14, IC₅₀: 4 nM	PARP15, IC₅₀: 4200 nM			99.29%
JW 55						TNKS1, IC₅₀: 1.9 μM	TNKS2, IC₅₀: 0.83 μM							99.83%
DPQ		PARP-1												99.68%
PJ34 hydrochloride	PARP, IC₅₀: 110 nM	PARP-1, IC₅₀: 110 nM	PARP-2, IC₅₀: 86 nM											99.81%
5,7,4'-Trimethoxyflavone	PARP													99.65%
DB008													PARP16, IC₅₀: 0.27 μM	98.47%
Gomisin N		PARP-1												99.94%
AZD-2461		PARP1, IC₅₀: 5 nM	PARP2, IC₅₀: 2 nM	PARP3, IC₅₀: 200 nM										99.79%
iRucaparib-AP6		PARP1, DC₅₀: 82 nM												99.03%
Venadaparib		PARP1, IC₅₀: 1.4 nM	PARP2, IC₅₀: 1 nM											98.11%
OM-153						TNKS1, IC₅₀: 13 nM	TNKS2, IC₅₀: 2 nM							99.30%
ME0328		ARTD1/PARP1, IC₅₀: 6.3 μM	ARTD2/PARP2, IC₅₀: 10.8 μM	ARTD3/PARP3, IC₅₀: 0.89 μM		ARTD5/TNKS1, IC₅₀: 47.3 μM	ARTD6/TNKS2, IC₅₀: 34.3 μM		ARTD10/PARP10, IC₅₀: 71.3 μM					99.64%
N-Descyclopropanecarbaldehyde Olaparib	PARP	PARP1	PARP-2											99.46%
RK-287107						tankyrase-1, IC₅₀: 14.3 nM	tankyrase-2, IC₅₀: 10.6 nM							99.80%
AZ6102		PARP1, IC₅₀: 2 μM	PARP2, IC₅₀: 0.5 μM			TNKS1, IC₅₀: 3 nM	TNKS2, IC₅₀: 2 nM							99.53%
MSC2504877		PARP1, IC₅₀: 0.54 μM												99.25%
1,5-Isoquinolinediol	PARP, IC₅₀: 0.18-0.37 μM													99.14%
Prostaglandin A2		PARP-1												99.9%
MN-64		ARTD1, IC₅₀: 19.1 μM	ARTD2, IC₅₀: 39.4 μM			TNKS1, IC₅₀: 6 nM	TNKS2, IC₅₀: 72 nM							99.61%
Sulfabenzamide		PARP1												99.68%
Niraparib tosylate hydrate		PARP-1, IC₅₀: 3.8 nM	PARP-2, IC₅₀: 2.1 nM	PARP-3, IC₅₀: 1300 nM	V-PARP, IC₅₀: 330 nM	TANK-1, IC₅₀: 570 nM								99.97%
Veliparib dihydrochloride		PARP-1, Ki: 5.2 nM	PARP-2, Ki: 2.9 nM											99.98%
Iniparib		PARP1												99.74%
CT-179	PARP													99.61%
7-Methylguanine		PARP-1, Ki: 61 μM												99.97%
PARP7-IN-15								PARP7, IC₅₀: 0.56 nM						99.03%
Nesuparib			PARP2, IC₅₀: 2 nM			tankyrase-1, IC₅₀: 5 nM	tankyrase-2, IC₅₀: 1 nM							99.54%
(8R,9S)-Talazoparib		PARP-1, IC₅₀: 144 nM												98.28%
PARP14 inhibitor H10										PARP14, IC₅₀: 490 nM				99.46%
PROTAC PARP1 degrader-1		PARP-1, DC₅₀: 252.5 nM												99.86%
PROTAC PARP1 degrader		PARP1												99.74%
BYK204165		hPARP-1, pIC₅₀: 7.35	mPARP-2, pIC₅₀: 5.38											99.89%
PARP1 PROTAC 180055		PARP1												98.90%
API-1	PARP													99.62%
NMS-P118		PARP-1, Kd: 9 nM	PARP-2, Kd: 1390 nM											99.54%
GeA-69										PARP14, Kd: 2.1 μM				99.91%
INO-1001	PARP													98.86%
KMR-206								PARP7, IC₅₀: 13.7 nM						98.86%
Niraparib (R-enantiomer)		PARP-1, IC₅₀: 2.4 nM												99.29%
PARP7-IN-16		PARP-1, IC₅₀: 0.94 nM	PARP-2, IC₅₀: 0.87 nM					PARP-7, IC₅₀: 0.21 nM						99.91%
5,7-Dihydroxychromone	PARP													99.94%
ASP3026		PARP1												99.88%
PARP10/15-IN-1									PARP10, IC₅₀: 160 nM		PARP15, IC₅₀: 370 nM
K-756						TNKS1, IC₅₀: 31 nM	TNKS2, IC₅₀: 36 nM							99.25%
PARP7-IN-16 free base		PARP1, IC₅₀: 0.94 nM	PARP2, IC₅₀: 0.87 nM					PARP7, IC₅₀: 0.21 nM						99.40%
PARP10-IN-3		human PARP1, IC₅₀: >100 μM	human PARP2, IC₅₀: 1.7 μM	human PARP3, IC₅₀: >100 μM	human PARP4, IC₅₀: 7 μM	human TNKS1, IC₅₀: 21 μM	human TNKS2, IC₅₀: 6.5 μM		human PARP10, IC₅₀: 480 nM	human PARP14, IC₅₀: 41 μM	human PARP15, IC₅₀: 1.7 μM	human PARP12, IC₅₀: >10 μM	human PARP16, IC₅₀: >10 μM	98.72%
RBN012811										PARP14, DC₅₀: 5 (KYSE-27 nM				98.79%
PARP1-IN-5 dihydrochloride		PARP-1, IC₅₀: 14.7 nM	PARP-2, IC₅₀: 0.9 μM
PARP7-IN-17								PARP7						99.81%
OUL312									PARP10					99.20%
PARP-1-IN-3		PARP-1, IC₅₀: 0.25 nM	PARP-2, IC₅₀: 2.34 nM											99.80%
PARPYnD		PARP1	PARP2											98.86%
PARP7-IN-22								PARP-7, IC₅₀: 0.6 nM						99.59%
A-620223		PARP-1, Ki: 8 nM												98.84%
PARP10/15-IN-3									PARP10, IC₅₀: 0.14 μM		PARP15, IC₅₀: 0.40 μM			99.23%
Simmiparib		PARP1, IC₅₀: 0.74 nM	PARP2, IC₅₀: 0.22 nM											99.01%
PARP1-IN-33		PARP1, IC₅₀: 0.41 nM												99.02%
A-966492		PARP-1, Ki: 1 nM	PARP-2, Ki: 1.5 nM											99.00%
Mefuparib hydrochloride		PARP1, IC₅₀: 3.2 nM	PARP2, IC₅₀: 1.9 nM			TNKS1, IC₅₀: 1.6 μM	TNKS2, IC₅₀: 1.3 μM							98.62%
KSQ-4279 gentisate		PARP1												99.75%
PARP10-IN-2		human PARP1, IC₅₀: >100 μM	human PARP2, IC₅₀: 27 μM	human PARP3, IC₅₀: >100 μM	human PARP4, IC₅₀: >100 μM	human TNKS1, IC₅₀: >100 μM	human TNKS2, IC₅₀: >100 μM		human PARP10, IC₅₀: 3.64 μM	human PARP14, IC₅₀: >100 μM	human PARP15, IC₅₀: 11 μM	human PARP12, IC₅₀: >10 μM	human PARP16, IC₅₀: >10 μM	98.02%
YCH1899		PARP-1, IC₅₀: <0.001 nM	PARP-2, IC₅₀: <0.001 nM	PARP3, IC₅₀: 1.1 nM	PARP4, IC₅₀: 1.0 nM	TNKS1, EC₅₀: 3.8 nM	TNKS2, IC₅₀: 12.4 nM	PARP-7, IC₅₀: 7.3 nM	ARTD10/PARP10, IC₅₀: 10.8 nM	PARP14, IC₅₀: 35.914 μM	PARP15, IC₅₀: 51.623 nM	human PARP12, IC₅₀: 14.1 nM		99.39%
PARP-1-IN-2		PARP-1, IC₅₀: 149 ± 11.0 nM												99.48%
PARP1-IN-11		PARP1, IC₅₀: 0.082 μM												99.42%
EB-47		ARTD1/PARP1, IC₅₀: 45 nM												99.89%
KU-0058948		PARP-1, IC₅₀: 3.4 nM												98.05%
NMS-P515		PARP-1, Kd: 16 nM PARP-1, IC₅₀: 27 nM (in Hela cells)												98.18%
PARP1-IN-29		PARP-1, IC₅₀: 6.3 nM
E7016	PARP													98.11%
TIQ-A			PARP2, IC₅₀: 210 nM				TNKS2, IC₅₀: 24 nM		PARP10, IC₅₀: >10 μM	PARP14, IC₅₀: >10 μM	PARP15, IC₅₀: 230 nM			99.85%
AZD-9574-acid		PARP-1												99.44%
PARP10/15-IN-2									PARP10, IC₅₀: 0.15 μM		PARP15, IC₅₀: 0.37 μM			98.92%
DR2313		PARP-1, IC₅₀: 0.20 μM	PARP-2, IC₅₀: 0.24 μM											99.66%
PARP-2-IN-1			PARP-2, IC₅₀: 11.5 nM											99.56%
PARP/PI3K-IN-1		PARP-1, pIC₅₀: 8.22	PARP-2, pIC₅₀: 8.44											99.40%
Procyanidin B2-3'-O-gallate	PARP
ART-IN-1			PARP2, IC₅₀: 19 μM				TNKS2, IC₅₀: 22 μM		PARP10, IC₅₀: 2.4 μM	PARP14, IC₅₀: >100 μM	PARP15, IC₅₀: 1.1 μM			98.91%
BPA-B9	PARP													98.50%
PROTAC PARP2 degrader-1			PARP-2, DC₅₀: 2 μM
Anticancer agent 43		PARP1												98.58%
PARP1/2/TNKS1/2-IN-1		PARP-1, IC₅₀: 0.25 nM	PARP-2, IC₅₀: 1.2 nM			TNKS1, IC₅₀: 13.5 nM	TNKS2, IC₅₀: 4.15 nM							98.66%
iVeliparib-AP6		PARP1, IC₅₀: 69 nM PARP1, ED₅₀: 36 nM	PARP2, IC₅₀: 21 nM PARP2, ED₅₀: 63 nM
KWZY-11		PARP1, IC₅₀: 156.8 nM	PARP2, IC₅₀: 197.3 nM
TNKS1/2-IN-1						TNKS1, pIC₅₀: 8.2 or 7.3	TNKS2, pIC₅₀: 7.1 or 7.7							99.24%
KU-0058684		PARP-1, IC₅₀: 3.2 nM
Rucaparib tartrate		PARP-1, Ki: 1.4 nM
Rucaparib camsylate		PARP-1, Ki: 1.4 nM
PARP1-IN-5		PARP-1, IC₅₀: 14.7 nM	PARP-2, IC₅₀: 0.9 μM
Venadaparib hydrochloride		PARP1, IC₅₀: 1.4 nM	PARP2, IC₅₀: 1 nM
Rucaparib acetate		PARP-1, Ki: 1.4 nM
Nesuparib hydrochloride			PARP2, IC₅₀: 2 nM			tankyrase-1, IC₅₀: 5 nM	tankyrase-2, IC₅₀: 1 nM
Rucaparib hydrochloride		PARP-1, Ki: 1.4 nM
PARP/VEGFR3-IN-1		PARP1, IC₅₀: 76.3 pM	PARP2, CC₅₀: 3.66 pM
2H-Indazole-7-carboxamide		PARP-1
AKT-IN-28	PARP
PARP1-IN-9		PARP1, IC₅₀: 30.51 nM
PARP-2-IN-3			PARP-2, IC₅₀: 0.07 μM
PARP1-IN-49		PARP1, IC₅₀: 23.56 nM PARP1, Kd: 17.78 nM	PARP2, IC₅₀: 285.39 nM
PARP1-IN-42		PARP-1, IC₅₀: <10 nM
PARP1/PKM2-IN-1		PARP1, IC₅₀: 39.5 nM
OM-1700						TNKS1, IC₅₀: 127 nM	TNKS2, IC₅₀: 14 nM
TOPOI/PARP-1-IN-2		PARP-1, IC₅₀: 32.2 nM	PARP-2, IC₅₀: 2844 nM
Antitumor agent-170								PARP7, IC₅₀: 7.05 nM
iRucaparib-TP3		PARP1, DC₅₀: 36 nM
PARP1/c-Met-IN-3		PARP1, IC₅₀: 3.7 nM	PARP2, IC₅₀: 4.52 nM
PARP1-IN-44		PARP1, IC₅₀: 0.6 nM	PARP2, IC₅₀: 1 nM	PARP3, IC₅₀: 12.5 nM		PARP5A, IC₅₀: 20.5 nM	PARP5B, IC₅₀: 38.1 nM	PARP7, IC₅₀: 7.5 nM
ARTD10/PARP10-IN-1		ARTD1/PARP1, IC₅₀: 4.4 μM							ARTD10/PARP10, IC₅₀: 0.8 μM	ARTD8/PARP14, IC₅₀: 1.6 μM	ARTD7/PARP15, IC₅₀: 1.7 μM
BER-IN-1		PARP-1
ZINC43120769		PARP1
ATR/PARP1-IN-1		PARP1, IC₅₀: 0.38 nM	PARP2, IC₅₀: 5.1 nM			TNKS1, IC₅₀: 116 nM	TNKS2, IC₅₀: 740.5 nM	PARP7, IC₅₀: 28.5 nM
PARP1/EZH2-IN-1		PARP-1, IC₅₀: 28 nM	PARP2, IC₅₀: 414 nM
PARP1/BRD4-IN-1		PARP1, IC₅₀: 49 nM
TC-E 5001						TNKS1, Ki: 79 nM	TNKS2, Ki: 28 nM
Bcl-2/Mcl-1-IN-5		PARP1
PARP1/CDK12-IN-1		PARP1, IC₅₀: 34 nM
YCH3292		PARP1, IC₅₀: <0.001 nM	PARP2, IC₅₀: <0.001 nM
PARP1-IN-47		PARP1, IC₅₀: <100 nM
PARP14 inhibitor 1				PARP3, IC₅₀: 2024 nM		PARP5A, IC₅₀: 1964 nM	PARP5B, IC₅₀: 1330 nM	PARP7, IC₅₀: 1973 nM	PARP10, IC₅₀: 5232 nM	PARP14, IC₅₀: 5.52 nM	PARP15, IC₅₀: 916 nM	human PARP12, IC₅₀: 3752 nM
PARP-1/2-IN-5		PARP-1, IC₅₀: 118 nM	PARP-2, IC₅₀: 11 nM
PARP1-IN-45		PARP1, IC₅₀: 17 nM
BWA-6047		PARP-1
DLC-50		PARP1, IC₅₀: 1.2 nM
(rac)-Talazoparib		PARP1, Ki: 1.2 nM	PARP2, Ki: 0.87 nM
PARP1-IN-8		PARP-1, IC₅₀: 97 nM												99.29%
EGFR-IN-197	PARP
AZ0108		PARP1, IC₅₀: 0.03 μM	PARP2, IC₅₀: 0.03 μM	PARP3, IC₅₀: 2.8 μM		TNKS1, IC₅₀: 3.2 μM
PARP7-IN-12								PARP7, IC₅₀: 7.836 nM
PARP/EZH2-IN-2		PARP1, IC₅₀: 6.89 ± 0.7 nM
DPQ hydrochloride		PARP-1
XW-17										PARP14
IDO1-IN-34		PARP-1
TNKS-IN-1		PARP-1, IC₅₀: >10000 nM				TNKS1, IC₅₀: 7.9 nM	TNKS2, IC₅₀: 8.7 nM
PARP1/BRD4-IN-2		PARP1, IC₅₀: 197 nM
Antitumor agent-214		PARP-1
TP-110	PARP
PARP1-IN-14		PARP1, IC₅₀: 0.6 ± 0.1 nM
Vrucaparib-TP4		PARP1
PARP1-IN-46		PARP-1, IC₅₀: 2.4 nM
PARP7-IN-23								PARP7
Tankyrase-IN-4						TNKS1, IC₅₀: 0.8 nM
PARP1-IN-21		PARP1
MC2050		PARP-1, IC₅₀: 119 nM	PARP-2, IC₅₀: 1.8 μM
PARP1-IN-43		PARP-1, IC₅₀: 5 nM
Anticancer agent 64	PARP
PARP1-IN-52		PARP-1
PC8		PARP1, IC₅₀: 0.126 μM
Lss-11		PARP1
Antitumor agent-169								PARP7, IC₅₀: 2.5 nM
PROTAC PARP1 degrader-5		PARP1, DC₅₀: 0.12 μM
TNKS-IN-4						TNKS1, IC₅₀: 0.1 nM	TNKS2, IC₅₀: 7.6 nM
Apoptosis inducer 45	PARP
TIPARP-IN-1								PARP7, IC₅₀: 2.15 nM
PARP1-IN-51		PARP1
PARP1-IN-37		PARP1, IC₅₀: 24 nM
Cathepsin-IN-5		PARP1
Tankyrase-IN-3						TNKS1, IC₅₀: 22 nM
NDs-IN-1		hPARP-1	PARP-2
PARP1 degrader 1		PARP-1, DC₅₀: 618 nM
KU-0058948 hydrochloride		PARP-1, IC₅₀: 3.4 nM
PARP1-IN-18		PARP1, IC₅₀: 2.7 nM
PARP1-IN-34		PARP1, IC₅₀: 0.32 nM	PARP2, IC₅₀: 326 nM
PARP/EZH2-IN-1		PARP-1, IC₅₀: 6.87 nM
PARP7-IN-24								PARP7
PARP1 degrader-2		PARP1, DC₅₀: 2.16 μM
PARP-1-IN-23		PARP-1, IC₅₀: 12.38 nM
PARP-2/1-IN-2		PARP1, Ki: 5 nM	PARP2, Ki: 2 nM
PARP7-IN-25								PARP7, IC₅₀: 1.582 nM
PARP1/NAMPT-IN-1		PARP1, IC₅₀: 1.2 nM
PARP1/BRD4-IN-3		PARP1, IC₅₀: 2019 nM
OUL245		PARP-1, IC₅₀: 570 nM	PARP2, IC₅₀: 44 nM	PARP3, IC₅₀: 8.8 μM	PARP4, IC₅₀: 6.0 μM	TNKS1, IC₅₀: 1.6 μM	TNKS2, IC₅₀: 370 μM		PARP10, IC₅₀: 2.9 μM	PARP14, IC₅₀: 6.7 μM	PARP15, IC₅₀: 2.0 μM
PARP1/c-Met-IN-1		PARP1, IC₅₀: 3.3 nM
EGFR/PARP-1-IN-1		PARP-1, IC₅₀: 12 nM
PARP1/ERK IN-1		PARP1, IC₅₀: 0.9 nM
PARP1-IN-22		PARP1
PROTAC FTO degrader 1		PARP1
PARP1-IN-10		PARP1, IC₅₀: 50.62 nM (^[1])
SK-575-NEG		PARP-1, IC₅₀: 2.64 nM
PARP1-IN-55		PARP1, IC₅₀: 0.019 μM
PARP14 inhibitor 2										PARP14, IC₅₀: <30 nM
PARP-1/HDAC-IN-1		PARP-1, IC₅₀: 68.90 nM
PARP1/2-IN-3		PARP-1, IC₅₀: 0.2235 nM
GPS167	PARP
13'-Carboxy-δ-tocopherol		PARP-1
UNPD139734		PARP-1
PARP1-IN-17		PARP-1
PARP-1/2/7-IN-1		PARP1	PARP2					PARP7
PARP1-IN-48		PARP1
MAPK-IN-5		PARP-1
PARP1-IN-30		PARP1
ARTD10/PARP10-IN-2		ARTD1/PARP1, IC₅₀: 9.7 μM							ARTD10/PARP10, IC₅₀: 2.0 μM	ARTD8/PARP14, IC₅₀: >20 μM	ARTD7/PARP15, IC₅₀: >20 μM
ZINC000081009201		PARP1, IC₅₀: 1.4767 μM
YCH3971		PARP-1, IC₅₀: 7.52 nM PARP-1, EC₅₀: 67.75 nM
PCIP-1			PARP2
PARP1-IN-20		PARP1, IC₅₀: 4.62 nM
PARP1-IN-50		PARP-1, IC₅₀: 64.98 nM
PARP1-IN-12		PARP-1, IC₅₀: 2.99 nM
TNKS-2-IN-4		PARP-1, IC₅₀: 860 nM				TNKS1, IC₅₀: 244 nM	TNKS2, IC₅₀: 19 nM
L-2286		PARP-1
PARP1-IN-35		PARP1, IC₅₀: 0.2 nM	PARP2, IC₅₀: 122 nM
PROTAC PARP1 degrader-3		PARP-1, DC₅₀: 58.14 nM
CEP-9722		PARP-1, IC₅₀: 20 nM	PARP-2, IC₅₀: 6 nM
PARP7-IN-21								PARP7
CDK9/PARP-IN-1		PARP1, IC₅₀: 107 nM
PARP10-IN-4						TNKS1, pIC₅₀: 6.95	TNKS2, pIC₅₀: 7.03		PARP10, pIC₅₀: 7.95
FLC-8	PARP
PARP1-IN-53		PARP-1, IC₅₀: 0.1 nM	PARP-2, IC₅₀: 23 nM
DDO3602		PARP1
2'-Nitroflavone		PARP1
PARP1/c-Met-IN-2		PARP1, IC₅₀: 21.8 nM
PARP10-IN-1									PARP10, IC₅₀: 1.8 or 2.7 μM
TNKS-2-IN-3		PARP1	PARP2			TNKS1	TNKS2
ST7710AA1		PARP-1, IC₅₀: 0.07 μM
8-Chloroquinazolin-4-ol		PARP-1, IC₅₀: 5.65 μM												98.44%
Benzo[c][1,8]naphthyridin-6(5H)-one		PARP-1, IC₅₀: 0.311 μM
BSI-401		PARP-1
UPF-1035		PARP-1, IC₅₀: 9 μM	PARP-2, IC₅₀: 0.15 μM
TNKS-IN-3							TNKS2, Ki: 8.5 nM
EXQ-2d						TNKS1, IC₅₀: 48.8 nM	TNKS2, IC₅₀: 13.8 nM
WD2000-012547		PARP-1, pKi: 8.221

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