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Cat. No.: HY-111501R

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H4R antagonist 1 (Standard)

H4R antagonist 1 (Standard) is the analytical standard of H4R antagonist 1 (HY-111501). This product is intended for research and analytical applications. H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC₅₀ of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R.

For research use only. We do not sell to patients.

CAS No.: 1429375-54-1
Formula: C₁₁H₁₁BrN₈
Molecular Weight:335.16

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

H4R antagonist 1 (Standard) Chemical Structure

CAS No.: 1429375-54-1

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Information

Application

The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.

Chemical Information

CAS No. 1429375-54-1
Molecular Weight 335.16
Formula C₁₁H₁₁BrN₈
SMILES

CNC(C1)CN1C2=NC3=NC=C(Br)C=C3N4C2=NN=N4
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Ko K, et al. Discovery of a Novel Highly Selective Histamine H4 Receptor Antagonist for the Treatment of Atopic Dermatitis. J Med Chem. 2018 Apr 12;61(7):2949-2961. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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