1429375-54-1
1429375-54-1
Chemical Structure
H4R antagonist 1
- CAS No.: 1429375-54-1
- Formula:C11H11BrN8
- Molecular Weight:335.16
IUPAC Name: 1-(8-bromopyrido[2,3-e]tetrazolo[1,5-a]pyrazin-4-yl)-N-methylazetidin-3-amine
InChIKey: ICGICUHMULRYIQ-UHFFFAOYSA-N
SMILES: CNC(C1)CN1C2=NC3=NC=C(Br)C=C3N4C2=NN=N4
Biological Activity: H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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H4R antagonist 1 | 99.82% | H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R. | ||||||||||||||||||||
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H4R antagonist 1 (Standard) | ≥98% | H4R antagonist 1 (Standard) is the analytical standard of H4R antagonist 1 (HY-111501). This product is intended for research and analytical applications. H4R antagonist 1 is a potent and highly selective histamine H4 receptor (H4R) antagonist with an IC50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R. | ||||||||||||||||||||
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