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Cat. No.: HY-186190

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I-FAPI-04 prodrug-1

I-FAPI-04 prodrug-1 is a prodrug of I-FAPI-04, which is an inhibitor targeting fibroblast activation protein (FAP). I-FAPI-04 prodrug-1 can be used as a radioactive tracer in cancer.

For research use only. We do not sell to patients.

CAS No.: 3032403-10-1
Formula: C₃₄H₄₀F₂N₆O₄Sn
Molecular Weight:753.43

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

I-FAPI-04 prodrug-1 Chemical Structure

CAS No.: 3032403-10-1

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- In Vivo
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

I-FAPI-04 prodrug-1 is a prodrug of I-FAPI-04, which is an inhibitor targeting fibroblast activation protein (FAP). I-FAPI-04 prodrug-1 can be used as a radioactive tracer in cancer^[1].

In Vivo

The active ingredient I-FAPI-04 of I-FAPI-04 prodrug-1 (Compound 8) significantly suppresses the tumor growth
in U87MG xenograft mice without significant toxicity^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 3032403-10-1
Molecular Weight 753.43
Formula C₃₄H₄₀F₂N₆O₄Sn
SMILES

O=C(N1[C@@H](CC(F)(C1)F)C#N)CNC(C2=CC=NC3=C2C=C(OCCCN4CCN(CC4)C(C5=CC=C(C=C5)[Sn](C)(C)C)=O)C=C3)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Ma H, et al. Synthesis and Preliminary Evaluation of ¹³¹I-Labeled FAPI Tracers for Cancer Theranostics. Mol Pharm. 2021;18(11):4179-4187. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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