Kv7.2/Kv7.3 agonist 1
Kv7.2/Kv7.3 agonist 1 (Compound 16) is an orally active agonist for KV7.2/7.3 channel (KCNQ2/3) with an EC50 of 1.03 μM. Kv7.2/Kv7.3 agonist 1 exhibits analgesic efficacy in mice chronic constriction injury (CCI) model and mice Streptozotocin (HY-13753)-induced diabetic peripheral neuropathic pain (DPNP) model, with ED50 of 12.02 and 9.63 mg/kg.
For research use only. We do not sell to patients.
- CAS No.: 2315450-35-0
- Formula: C14H14FN3O2
- Molecular Weight:275.28
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
KCNQ2/Q3 1.03 μM (EC50) |
Chemical Information
-
CAS No. 2315450-35-0
-
Molecular Weight 275.28
-
Formula C14H14FN3O2
-
SMILES
CC(NC1=NC(OCC2=CC=C(F)C=C2)=CC=C1N)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Kv7.2/Kv7.3 agonist 1 Related Classifications
HY-168214 Related Classifications
Powered by Bioz