2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. KY 234

KY 234 is an orally effective inhibitor that targets thromboxane A2 production, with an IC50 of 5 μM. KY 234 significantly inhibits leukotriene D4 (LTD4), histamine, and antigen-induced bronchoconstriction in guinea pigs, with IC50 values of 6.0 mg/kg, 2.5 mg/kg, and 6.3 mg/kg, respectively.

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KY 234

KY 234 Estructura química

No. CAS : 172544-75-1

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KY 234 Related Antibodies

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Descripciòn

KY 234 is an orally effective inhibitor that targets thromboxane A2 production, with an IC50 of 5 μM. KY 234 significantly inhibits leukotriene D4 (LTD4), histamine, and antigen-induced bronchoconstriction in guinea pigs, with IC50 values of 6.0 mg/kg, 2.5 mg/kg, and 6.3 mg/kg, respectively[1].

IC50 & Target

Thromboxane A2 receptor[1]
Peso molecular

555.65

Fòrmula

C33H34N5NaO2
No. CAS
SMILES

O=C(C1=CC2=C(C=C1)C(CN3C=CN=C3)=CN2CCCN4CCN(C(C5=CC=CC=C5)C6=CC=CC=C6)CC4)O[Na]
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.
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Referencias
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KY 234 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

KY 234172544-75-1KY234KY-234Histamine ReceptorInhibitorinhibitorinhibit

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Nombre del producto:
KY 234
Cat. No.:
HY-117842
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