1 Result for "

μOR/σ1R

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "μOR/σ1R" in MCE Product Catalog:

Cat. No.: HY-163065
CAS No.: 3009018-61-2
Research Areas:  

Neurological Disease

σ1 Receptor/μ Opioid receptor modulator 2 (compound 4x) is a dual μOR agonist/σ1R antagonist, and displays picomolar μOR agonism activity (EC50: 0.6 ± 0.2 nM) and good σ1R inhibitory activity (Ki: 363.7 ± 5.6 nM). σ1 Receptor/μ Opioid receptor modulator 2 exhibits robust analgesic effects in various pain models .
loading...
    loading...