1 Result for "

JAK2-IN-7

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "JAK2-IN-7" in MCE Product Catalog:

Cat. No.: HY-131906
CAS No.: 2593402-36-7
Purity:  99.15%
Target:  

JAK FLT3 Apoptosis

Research Areas:  

Cancer

JAK2-IN-7 is a selective JAK2 inhibitor with IC50s of 3, 11.7, and 41 nM for JAK2, SET-2, and Ba/F3 V617F cells, respectively. JAK2-IN-7 possesses >14-fold selectivity over JAK1, JAK3, FLT3. JAK2-IN-7 stimulates cell cycle arrest in the G0/G1 phase and induces tumor cellapoptosis. Antitumor activities .
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