88 Results for "

Pentapeptide

" in MedChemExpress (MCE) Product Catalog:
Products (88)

88 Results for "Pentapeptide" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-P0288
CAS No.: 58822-25-6
Synonyms: Leu-enkephalin; Leucine enkephalin; Leucyl-enkephalin
[Leu5]-Enkephalin is a pentapeptide with morphine like properties. [Leu5]-Enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.
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2
2 Cited Publications
Cat. No.: HY-19884B
CAS No.: 2863659-22-5
Synonyms: RM-131 TFA; BIM-28131 TFA
Target:  

GHSR

Research Areas:  

Metabolic Disease

Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin TFA is centrally penetrant. Relamorelin TFA increases growth hormone levels and accelerates gastric emptying. Relamorelin TFA has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research .
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2
2 Cited Publications
Cat. No.: HY-N8395
CAS No.: 66054-36-2
Synonyms: Tunicamycin A
Tunicamycin V (Tunicamycin A) is a nucleoside natural product that inhibits bacterial phospho-N-acetylmuramyl-pentapeptide transferase (MraY) with an IC50 of 0.35?μM. Tunicamycin V has antibacterial activties .
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1
1 Cited Publications
Cat. No.: HY-16485
CAS No.: 560130-42-9
Synonyms: TD-6424 hydrochloride
Target:  

Antibiotic Bacterial

Research Areas:  

Infection

Telavancin hydrochloride (TD-6424 hydrochloride) is a bactericidal agent that exhibits inhibitory activity against Staphylococcus aureus. Telavancin hydrochloride inhibits bacterial cell wall synthesis by binding to the lipid-linked N-acetylglucosamine-N-muramyl pentapeptide (with a D-Ala-D-Ala terminus), a peptidoglycan precursor, and blocks the transglycosylation and transpeptidation steps. Telavancin hydrochloride disrupts bacterial membrane barrier function, induces dissipation of bacterial membrane potential, and causes leakage of cytoplasmic ATP and potassium ions, with its activity restricted exclusively to bacterial membranes. Telavancin hydrochloride can be used in research on bacterial infections, central venous catheter-related bloodstream infections, and Gram-positive bacterial pneumonia .
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1
1 Cited Publications
Cat. No.: HY-P5919
CAS No.: 2614-55-3
Target:  

Peptides

Research Areas:  

Others

Ala-D-γ-Glu-Lys-D-Ala-D-Ala is the pentapeptide tail of the peptidoglycan precursor UDPMurNAc-l-Ala-γ-d-Glu-l-Lys(Gly)(5)-d-Ala-d-Ala .
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1
1 Cited Publications
Cat. No.: HY-P0275
CAS No.: 57966-42-4
Proctolin is an endogenous pentapeptide that acts as an excitatory neuromodulator.
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Cat. No.: HY-P0045
CAS No.: 214047-00-4
Synonyms: Matrixyl; Palmitoyl Pentapeptide 3; Matrixyl (Palmitoyl Pentapeptide)
Target:  

Collagen

Research Areas:  

Others

Palmitoyl pentapeptide 4 (Matrixyl; Palmitoyl pentapeptide 3; Matrixyl (Palmitoyl Pentapeptide) is a bioactive peptide with anti-ageing effect and has been reported used as a cosmetic ingredient [1]
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Cat. No.: HY-33046
CAS No.: 120205-50-7
Synonyms: (2R,3R)-BOC-dolaproine
Research Areas:  

Cancer

N-Boc-dolaproine ((2R,3R)-BOC-dolaproine) is the amino acid residue of the pentapeptide Dolastatin 10 (HY-15580). Dolastatin 10 inhibits tubulin polymerization and mitosis and has anticancer activity .
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Cat. No.: HY-138053
CAS No.: 90831-71-3
Synonyms: Ristomycin III
Target:  

Antibiotic

Research Areas:  

Cardiovascular Disease Infection

Ristocetin A sulfate (Ristomycin III) is a glycopeptide antibiotic that binds to von Willebrand factor (VWF) and bacterial cell wall components. Ristocetin A sulfate interferes with the biosynthesis of bacterial peptidoglycan by inhibiting transpeptidation. As an inducer of platelet adhesion and aggregation, Ristocetin A sulfate drives conformational changes by binding to the A1 domain of VWF, thereby activating downstream signaling pathways and promoting cytoskeletal rearrangement. Ristocetin A sulfate not only enhances platelet adhesion and spreading on immobilized VWF, but also induces the formation of asymmetric dimers with anticooperativity between platelets and plasma VWF. Ristocetin A sulfate is widely used in studies related to thromboembolic diseases and bacterial infections .
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Cat. No.: HY-P0099
CAS No.: 135679-88-8
Target:  

nAChR

Research Areas:  

Others

Pentapeptide-3 is a pentapeptide fragment of neurotoxin waglerin-1, it can be extracted from the venom of Temple Viper. Pentapeptide-3 is a competitive antagonist of nicotinic acetylcholine receptors (nAChRs), it can blocks nerves at the post-synaptic membrane. Pentapeptide-3 has anti-aging effects and it can be used together with other cosmetic peptides .
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Cat. No.: HY-107024
CAS No.: 105250-85-9
Purity:  99.77%
Synonyms: OGP(10-14); Historphin
Target:  

Src

Research Areas:  

Others

Osteogenic Growth Peptide (10-14) (OGP(10-14)), the C-terminal truncated pentapeptide of osteogenic growth peptide (OGP), retains the full OGP-like activity. Osteogenic Growth Peptide (10-14) is responsible for the binding to the OGP receptor and activates an intracellular Gi-protein-MAP kinase signaling pathway. Osteogenic Growth Peptide (10-14) is a potent mitogen and stimulator of osteogenesis and hematopoiesis. Osteogenic Growth Peptide (10-14) acts as a Src inhibitor .
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Cat. No.: HY-P0295
CAS No.: 96426-21-0
Synonyms: GRGDS
Target:  

Integrin

Research Areas:  

Others

Gly-Arg-Gly-Asp-Ser (GRGDS) is a pentapeptide that forms the cell-binding domain of a glycoprotein, osteopontin. Gly-Arg-Gly-Asp-Ser binds to integrin receptors αvβ3 and αvβ5 with estimated IC50 of ~5 and ~6.5 μM
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Cat. No.: HY-105077A
CAS No.: 204992-09-6
Purity:  98.01%
Synonyms: INN 00835 diTFA
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Nemifitide diTFA (INN 00835 diTFA) is a synthetic pentapeptide antidepressant with a potential for rapid onset of action . Nemifitide diTFA is a peptide analog of melanocyte-inhibiting factor (MIF) . Nemifitide diTFA can cross the blood-brain barrier .
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Cat. No.: HY-P5840
CAS No.: 1206475-79-7
Research Areas:  

Cancer

Cyclo(RGDyC) is a cyclic pentapeptide with anti-angiogenic abilities. Cyclo(RGDyC) can be combined with liposome delivery systems for research on ocular neovascular diseases and cancer .
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Cat. No.: HY-P4102
CAS No.: 1810853-35-0
Target:  

Peptides

Research Areas:  

Cancer

Cyclic PSAP peptide is a cyclic pentapeptide (DWLPK). Cyclic PSAP peptide exhibits agent-like properties and could inhibit metastatic spread and restrain tumor development in general in vivo .
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Cat. No.: HY-P4047
CAS No.: 1228992-90-2
Target:  

Drug Derivative

Research Areas:  

Others

Cyclo(RGDfK(Mal)) is a pentapeptide. Cyclo(RGDfK(Mal)) improves the attachment and infiltration of human pluripotent stem cells. Cyclo(RGDfK(Mal)) can be used for 3D stem cell culture and expansion .
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Cat. No.: HY-P10641A
Target:  

Peptides

Research Areas:  

Cardiovascular Disease

Heart-homing peptide TFA is a Pentapeptide, CRPPR. CRPPR is a linear peptide containing arginine that has been identified as a heart-homing peptide owing to its ability to specifically bind to heart endothelium, and cysteine-rich protein-2 (CRIP-2) has been proposed as the receptor. Heart-homing peptide TFA can be used for conjugating liposomes .
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Cat. No.: HY-P0103A
CAS No.: 2763588-80-1
Target:  

LPL Receptor

Research Areas:  

Metabolic Disease

Myristoyl pentapeptide-17 acetate can stimulate eyelash growth by stimulating keratin production. Myristoyl pentapeptide-17 acetate promotes the delivery of key ingredients in the serum, such as the growth factors and lysophosphatidic acid .
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Cat. No.: HY-P0103
CAS No.: 959610-30-1
Target:  

LPL Receptor

Research Areas:  

Metabolic Disease

Myristoyl pentapeptide-17 can stimulate eyelash growth by stimulating keratin production. Myristoyl pentapeptide-17 promotes the delivery of key ingredients in the serum, such as the growth factors and lysophosphatidic acid .
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Cat. No.: HY-P5239
CAS No.: 1392416-25-9
Target:  

Collagen

Research Areas:  

Others

Myristoyl pentapeptide-4 is a bioactive peptide with promotion of hair growth effect and has been reported used as a cosmetic ingredient .
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