4 Results for "

Tyr385

" in MedChemExpress (MCE) Product Catalog:
Products (4)

4 Results for "Tyr385" in MCE Product Catalog:

Methylhydroquinone
Methylhydroquinone
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Cat. No.: HY-W012817
CAS No.: 95-71-6
Category:  

Natural Products Microorganisms Other Diseases Disease Research Fields

Target:  

Environmental Pollutants COX

Methylhydroquinone is an orally active COX inhibitor with IC50s of 480.7 μM and 52.2 μM for ovine COX-1 and human recombinant COX-2, respectively. Methylhydroquinone has potential DNA damaging effects: 1) inhibiting COX-1 to reduce prostaglandin synthesis and exert anti-inflammatory activity; 2) inducing DNA single-strand breaks. Methylhydroquinone exerts its effects by competitively binding to the active sites of COX-1 (such as Tyr385, Met522) and non-covalent interactions .
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Plipastatin A1
Plipastatin A1
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Cat. No.: HY-P10447
CAS No.: 103651-09-8
Synonyms: Fengycin IX; SNA-60-367-3
Target:  

Phospholipase Fungal

Research Areas:  

Infection

Plipastatin A1 (Fengycin IX; SNA-60-367-3) is a lipopeptide with phospholipase A2 inhibitory activity. Plipastatin A1 inhibits conidial germination of Botrytis cinerea in vitro and reduces the incidence of gray mold on tomato leaves. Plipastatin A1 is applicable to research related to gray mold [1][2].
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Methylhydroquinone (Standard)
Methylhydroquinone (Standard)
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Cat. No.: HY-W012817R
CAS No.: 95-71-6
Category:  

Natural Products Microorganisms

Target:  

COX Reference Standards

Methylhydroquinone (Standard) is the analytical standard of Methylhydroquinone. This product is intended for research and analytical applications. Methylhydroquinone is an orally active COX inhibitor with IC50s of 480.7 μM and 52.2 μM for ovine COX-1 and human recombinant COX-2, respectively. Methylhydroquinone has potential DNA damaging effects: 1) inhibiting COX-1 to reduce prostaglandin synthesis and exert anti-inflammatory activity; 2) inducing DNA single-strand breaks. Methylhydroquinone exerts its effects by competitively binding to the active sites of COX-1 (such as Tyr385, Met522) and non-covalent interactions[1][2].
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7-Methoxy-4H-chromen-4-one-o-carborane
7-Methoxy-4H-chromen-4-one-o-carborane
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Cat. No.: HY-183188
CAS No.: 3097646-97-1
Target:  

Androgen Receptor COX

Research Areas:  

Infection Neurological Disease Metabolic Disease Inflammation/Immunology Cancer

7-Methoxy-4H-chromen-4-one-o-carborane is an ER agonist and COX inhibitor with a COX-1 IC50 of 3.0 μM, COX-2 IC50 of 1.0 μM. 7-Methoxy-4H-chromen-4-one-o-carborane can be used for research on antimicrobial, anti-inflammatory, antitumor, neuroprotective, and estrogenic effects .
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