1. GPCR/G Protein
  2. Adenosine Receptor
  3. Arotinolol

Arotinolol 

Cat. No.: HY-122537A
Handling Instructions

Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol is an antihypertensive agent for the treatment of a variety of cardiovascular pathologies as well as non-cardiovascular diseases.

For research use only. We do not sell to patients.

Arotinolol Chemical Structure

Arotinolol Chemical Structure

CAS No. : 68377-92-4

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 74 In-stock
Estimated Time of Arrival: December 31
5 mg USD 90 In-stock
Estimated Time of Arrival: December 31
10 mg USD 150 In-stock
Estimated Time of Arrival: December 31
25 mg USD 330 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol is an antihypertensive agent for the treatment of a variety of cardiovascular pathologies as well as non-cardiovascular diseases[1].

IC50 & Target

IC50: α/β-adrenergic receptor

In Vivo

Arotinolol (oral gavage; 200 mg/kg; 8 weeks) can significantly decrease central arterial pressure (CAP) and pulse wave velocity (PWV), in addition, it reduces aortic collagen depositions and finally improves arterial stiffness in SHR mouse[1].

Animal Model: SHR mice[1]
Dosage: 200 mg/kg
Administration: Orally gavage; 200 mg/kg; once daily; 8 weeks
Result: Improved arterial stiffness in SHR.
Molecular Weight

371.54

Formula

C₁₅H₂₁N₃O₂S₃

CAS No.

68377-92-4

SMILES

O=C(C1=CC=C(C2=CSC(SCC(O)CNC(C)(C)C)=N2)S1)N

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

ArotinololAdenosine ReceptorP1 receptorhypertensionheart failuremyocardial infarctionischemic cardiac eventInhibitorinhibitorinhibit

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Arotinolol
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