(S)-GNE-987
(S)-GNE-987 (compound 4), the GNE-987 (a chimeric BET degrader) hydroxy-proline epimer, abrogates binding to von Hippel-Lindau and does not degrade BRD4 protein. (S)-GNE-987 can be used to design PROTAC-Antibody Conjugate (PAC).
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2738533-33-8
- Fòrmula: C56H67F2N9O8S2
- Peso molecular:1096.31
-
Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Actividad biológica
-
Chemical Information
- Pureza y Documentación
- Referencias
-
Help & FAQs
Ver todos los productos específicos de isoformas PROTACs
More
Actividad biológica
(S)-GNE-987 displays potent anti-MYC activity with an IC50 of 0.48 nM[1].
Chemical Information
-
No. CAS 2738533-33-8
-
Peso molecular 1096.31
-
Fòrmula C56H67F2N9O8S2
-
SMILES
O=C([C@H](C[C@H](O)C1)N1C([C@@H](NC(CCCCCCCCCCNC(C2=C(CS(=O)(C)=O)C=C(C(N(C3=NC=C(F)C=C3F)C4)=C2)C5=CN(C)C(C6=C5C4=CN6)=O)=O)=O)C(C)(C)C)=O)NCC7=CC=C(C(SC=N8)=C8C)C=C7
-
Envío
Room temperature in continental US; may vary elsewhere.
-
Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
(S)-GNE-987 Related Classifications
HY-129937 Related Classifications
Powered by Bioz