GIPR/GLP-1R/GCGR agonist-1
GIPR/GLP-1R/GCGR agonist-1 (compound 686) is a triple receptor agonist with activity at GLP-1R, GIPR, and GCGR. GIPR/GLP-1R/GCGR agonist-1 functionally modulates target receptors to drive cAMP generation. GIPR/GLP-1R/GCGR agonist-1 can be used for the research of type 2 diabetes mellitus, obesity, nonalcoholic fatty liver disease.
For research use only. We do not sell to patients.
- Formula: C238H360FN51O75
- Molecular Weight:5154.70
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Description
IC50 & Target
[1]|
GLP-1 |
Chemical Information
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Molecular Weight 5154.70
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Formula C238H360FN51O75
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Sequence
Tyr-{Aib}-Gln-Gly-Thr-{αMe-Phe(2F)}-Thr-Ser-Asp-{4Pal}-Ser-Ile-{αMe-Leu}-Leu-Asp-{Orn}-{Lys((y-Glu)2-CO-(CH2)16-COzH)}-Ala-Gln-{Me-4Pal}-{Orn}-Phe-Ile-{d-Glu}-{αMe-Tyr}-Leu-Ile-Glu-Gly-Gly-Pro-Ser-Ser-Gly-Glu-Pro-Pro-Pro-Glu-Thr-Glu-NH2
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Sequence Shortening
Y-{Aib}-QGT-{αMe-Phe(2F)}-TSD-{4Pal}-SI-{αMe-Leu}-LD-{Orn}-{Lys((y-Glu)2-CO-(CH2)16-COzH)}-AQ-{Me-4Pal}-{Orn}-FI-{d-Glu}-{αMe-Tyr}-LIEGGPSSGEPPPETE-NH2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)