Glucagon receptor antagonist-5
Glucagon receptor antagonist-5 (compound 13K) is a potent and orally bioavailable indazole-based glucagon receptor antagonist (Ki=32 nM). Glucagon receptor antagonist-5 has potential for the treatment of type 2 diabetes mellitus (T2DM).
For research use only. We do not sell to patients.
- CAS No.: 2200274-63-9
- Formula: C30H29ClF3N3O3
- Molecular Weight:572.02
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Ki: 32 nM (glucagon receptor)[1]
Chemical Information
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CAS No. 2200274-63-9
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Molecular Weight 572.02
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Formula C30H29ClF3N3O3
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SMILES
O=C(NCCC(O)=O)C1=CC=C([C@@H](N2N=CC3=C2C=C(C)C(C4=CC=C(C(F)(F)F)C=C4Cl)=C3)CC(C)C)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)