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Cat. No.: HY-101340AR

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Luvixasertib hydrochloride (Standard)

(Synonyms: CFI-402257 hydrochloride (Standard))

Luvixasertib (hydrochloride) (Standard) is the analytical standard of Luvixasertib (hydrochloride) (HY-101340A). This product is intended for research and analytical applications. CFI-402257 hydrochloride is a highly selective and orally bioavailable TTK/Mps1 inhibitor with an IC50 of 1.7 nM for TTK in vitro. CFI-402257 hydrochloride has anti-cancer activity.

For research use only. We do not sell to patients.

CAS No.: 1610677-37-6
Formula: C₂₈H₃₁ClN₆O₃
Molecular Weight:535.04

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Luvixasertib hydrochloride (Standard) Chemical Structure

CAS No.: 1610677-37-6

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Application

The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.

Chemical Information

CAS No. 1610677-37-6
Molecular Weight 535.04
Formula C₂₈H₃₁ClN₆O₃
SMILES

CC1=CC(C2=C3N=C(OC4=CN=CC=C4)C=C(NC[C@@H]5C[C@@](O)(C)C5)N3N=C2)=CC=C1C(NC6CC6)=O.Cl
Synonyms

CFI-402257 hydrochloride (Standard)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

References

[1]. Liu Y, et al. Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer Agent. ACS Med Chem Lett. 2016 May 6;7(7):671-5. [Content Brief]

[2]. Mason JM, et al. Functional characterization of CFI-402257, a potent and selective Mps1/TTK kinase inhibitor, for the treatment of cancer. Proc Natl Acad Sci U S A. 2017 Mar 21;114(12):3127-3132. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Luvixasertib hydrochloride (Standard)

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Luvixasertib hydrochloride (Standard)

Product Information

Chemical Information

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References

Calculators

Help & FAQs

Luvixasertib hydrochloride (Standard) Related Classifications

HY-101340AR Related Classifications