3 Results for "

1354799-87-3

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "1354799-87-3" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-19631
CAS No.: 1354799-87-3
Synonyms: NS-018 maleate
Target:  

JAK

Research Areas:  

Cancer

Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable JAK2 inhibitor, with an IC50 of 0.72 nM, 46-, 54-, and 31-fold selectivity for JAK2 over JAK1 (IC50, 33 nM), JAK3 (IC50, 39 nM), and Tyk2 (IC50, 22 nM).
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1
1 Cited Publications
Cat. No.: HY-19631A
CAS No.: 1239358-86-1
Synonyms: NS-018
Target:  

JAK

Research Areas:  

Cancer

Ilginatinib (NS-018) is a highly active and orally bioavailable JAK2 inhibitor, with an IC50 of 0.72 nM, 46-, 54-, and 31-fold selectivity for JAK2 over JAK1 (IC50, 33 nM), JAK3 (IC50, 39 nM), and Tyk2 (IC50, 22 nM).
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1
1 Cited Publications
Cat. No.: HY-19631B
CAS No.: 1239358-85-0
Synonyms: NS-018 hydrochloride
Target:  

JAK

Research Areas:  

Cancer

Ilginatinib hydrochloride (NS-018 hydrochloride) is a highly active and orally bioavailable JAK2 inhibitor, with an IC50 of 0.72 nM, 46-, 54-, and 31-fold selectivity for JAK2 over JAK1 (IC50, 33 nM), JAK3 (IC50, 39 nM), and Tyk2 (IC50, 22 nM).
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