1 Result for "

Cytosolic calcium flux

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "Cytosolic calcium flux" in MCE Product Catalog:

Cat. No.: HY-146401
CAS No.: 2304750-68-1
Target:  

CXCR

Research Areas:  

Cancer

CXCR4 antagonist 6 (compound 46) is a potent CXCR4 antagonist with an IC50 value of 79 nM. CXCR4 antagonist 6 inhibits CXCL12 induced cytosolic calcium flux (IC50 = 0.25 nM). CXCR4 antagonist 6 significantly mitigates CXCL12/CXCR4 mediated cell migration. CXCR4 antagonist 6 exhibits marked efficacy in a cancer metastasis model in mice .
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