2 Results for "

Thiazinamium

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Thiazinamium" in MCE Product Catalog:

14
14 Cited Publications
Cat. No.: HY-108896
CAS No.: 138614-30-9
Purity:  99.85%
Synonyms: HOE 140 acetate
Target:  

Bradykinin Receptor

Research Areas:  

Inflammation/Immunology

Icatibant acetate (HOE-140 acetate) is a potent and specific peptide antagonist of bradykinin B2 receptor with an IC50 and Ki of 1.07 nM and 0.798 nM respectively .
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Cat. No.: HY-U00267
CAS No.: 4320-13-2
Target:  

Cholinesterase (ChE)

Research Areas:  

Inflammation/Immunology

Thiazinamium (chloride) possesses potent anticholinergic and antiallergic activity and inhibits TxB2 synthesis with IC50 value of 0.2 µM. Thiazinamium (chloride) is structurally similar to H-1 antagonists Promethazine (HY-B1296). Thiazinamium (chloride) stimulates the phosphatidylcholine secretion in adult rat type II pneumocytes .
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