Sigma-2 Radioligand 1
Sigma-2 Radioligand 1 (compound 1) is a Sigma-2 selective ligand. Sigma-2 Radioligand 1 has good biodistribution in mice and good in vivo activity in rats. [18F] Modified Sigma-2 Radioligand 1 for visualization of tumors in micro-PET/CT imaging, exhibiting high tumor uptake and tumor-to-background ratio. Experiments show that Sigma-2 Radioligand 1 binds highly specifically in U87MG glioma xenografts.
For research use only. We do not sell to patients.
- CAS No.: 2860554-32-9
- Formula: C24H30FN3O3
- Molecular Weight:427.51
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
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Biological Activity
Ki: 2.57 nM (Sigma-2, σ2)[1]
Chemical Information
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CAS No. 2860554-32-9
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Molecular Weight 427.51
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Formula C24H30FN3O3
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SMILES
FCCN1C(N(C2=C1C=CC=C2)CCCCN3CCC4=C(C3)C=C(C(OC)=C4)OC)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Sigma-2 Radioligand 1 Related Classifications
HY-156124 Related Classifications
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