σ1 Receptor ligand 1
σ1 Receptor ligand 1 (compound 5I) is a σ1 receptor ligand with a Ki of 3.9 nM. σ1 Receptor ligand 1 has a high plasma protein binding (89%) and promising metabolic stability in the presence of mouse liver microsomes and NADPH. σ1 Receptor ligand 1 can be utilized in neurological and cancer research.
For research use only. We do not sell to patients.
- Formula: C22H28N2O2
- Molecular Weight:352.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Sigma Receptor Isoforms
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Biological Activity
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σ1 3.9 nM (Ki) |
Chemical Information
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Molecular Weight 352.47
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Formula C22H28N2O2
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SMILES
COC1=CC=C(C=C1)C2CCOC3(C2)CCN(CC3)CC4=CN=CC=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)