2. Signaling Pathways
  3. Epigenetics
  4. Histone Methyltransferase
  5. EZH1 Isoform
  6. EZH1 Inhibitor

EZH1 Inhibitor

EZH1 Inhibitors (3):

Cat. No. Product Name Effect Purity
  • HY-109108A
    Valemetostat tosylate
    		Inhibitor 98.14%
    Valemetostat (DS-3201) tosylate, a first-in-class EZH1/2 dual inhibitor with IC50 values ＜10 nM.
  • HY-109108
    Valemetostat
    		Inhibitor 99.65%
    Valemetostat (DS-3201), a first-in-class EZH1/2 dual inhibitor with IC50 values ＜10 nM.
  • HY-144881
    (S)-HH2853
    		Inhibitor
    (S)-HH2853 (compound 200), a PYRIDINO five membered aromatic ring compound, is a potent EZH1/2 dual inhibitor with an IC50 of <100 nM for EZH2_Y641F.