1. Signaling Pathways
  2. Epigenetics
    TGF-beta/Smad
  3. PKC
  4. PKC Inhibitors

PKC Inhibitors

PKC

PKCα

PKCβ

PKCγ

PKCδ

PKCε

PKCη

PKCζ

PKCθ

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform PKC together.

Please try each isoform separately.

PKC Specific Inhibitors, Antagonists & Activators
Product Name PKC PKCα PKCβ PKCγ PKCε PKC Selectivity Purity
Fasudil Hydrochloride
PKC, IC50: 12.30 μM
        Selective Inhibitor 99.91%
Fasudil
PKC, IC50: 12.3 μM
        Selective Inhibitor
Bisindolylmaleimide X hydrochloride
PKC
        Selective Inhibitor 98.53%
KT5823
PKC, Ki: 4 μM
        Selective Inhibitor
Phorbol 12-myristate 13-acetate
PKC, EC50: 11.7 nM
        Pan Activator 99.66%
Staurosporine
PKC, IC50: 6 nM
        Pan Inhibitor 99.98%
Bisindolylmaleimide I
Bovine brain PKC, IC50: 10 nM
PKCα, IC50: 20 nM
PKCβII, IC50: 16 nM
PKCβI, IC50: 17 nM
PKCγ, IC50: 20 nM
  Pan Inhibitor 98.14%
Mitoxantrone
PKC, IC50: 8.5 μM
        Pan Inhibitor >98.0%
Ro 31-8220 mesylate
Rat Brain PKC, IC50: 23 nM
PKC-α, IC50: 5 nM
PKC-βI, IC50: 24 nM
PKC-βII, IC50: 14 nM
PKC-γ, IC50: 27 nM
PKC-ε, IC50: 24 nM
Pan Inhibitor 99.28%
Mitoxantrone dihydrochloride
PKC, IC50: 8.5 μM
        Pan Inhibitor 98.01%
Valrubicin
TPA-activated PKC, IC50: 0.85 μM
PDBu-activated PKC, IC50: 1.25 μM
        Pan Inhibitor 99.95%
HA-100
PKC, IC50: 12 μM
PKC, Ki: 6.5 μM
        Pan Inhibitor 99.76%
TPPB
PKC, Ki: 11.9 nM
        Pan Activator 99.81%
Verbascoside
PKC, IC50: 25 μM
        Pan Inhibitor 99.61%
Ingenol
PKC, Ki: 30 μM
        Pan Activator >99.0%
CGP60474
PKC
        Pan Inhibitor 99.88%
Daphnetin
PKC, IC50: 25.01 μM
        Pan Inhibitor 99.55%
TAS-301
PKC
        Pan Inhibitor 99.50%
D-erythro-Sphingosine
PKC
        Pan Inhibitor >98.0%
Chelerythrine
PKC, IC50: 0.7 μM
        Pan Antagonist