PKC Activator

PKC Activators (28):

Cat. No.	Product Name	Effect	Purity

HY-18739

Phorbol 12-myristate 13-acetate	Activator	99.66%
Phorbol 12-myristate 13-acetate (PMA), a phorbol ester, is a dual SphK and protein kinase C (PKC) activator.

HY-13434

Ionomycin	Activator	≥99.0%
Ionomycin (SQ23377) is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus.

HY-13434A

Ionomycin calcium	Activator	≥98.0%
Ionomycin calcium (SQ23377 calcium) is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus.

HY-18985

Phorbol 12,13-dibutyrate	Activator	98.78%
Phorbol 12,13-dibutyrate (Phorbol dibutyrate) is a PKC activator and a potent skin tumor promoter.

HY-12307

(-)-Indolactam V	Activator	99.30%
(-)-Indolactam V is a PKC activator, with K_is of 3.36 nM, 1.03 μM for η-CRD2 (PKCη surrogate peptide), γ-CRD2 (PKCγ surrogate peptide), and K_ds of 5.5 nM (η-C1B), 7.7 nM (ε-C1B), 8.3 nM (δ-C1B), 18.9 nM (β-C1A-long), 20.8 nM (α-C1A-long), 137 nM (β-C1B), 138 nM (γ-C1A), 213 nM (γ-C1B), and has antitumor activity.

HY-108355

R59949	Activator	≥99.0%
R59949 is a pan diacylglycerol kinase (DGK) inhibitor with an IC₅₀ of 300 nM.

HY-18981

Decursin	Activator	99.94%
Decursin ((+)-Decursin) is a potent anti-tumor agent.

HY-12359

TPPB	Activator	99.81%
TPPB is a cell-permeable benzolactam-derived protein kinase C (PKC) activator with a K_i of 11.9 nM.

HY-107613

R 59-022	Activator	99.82%
R 59-022 (DKGI-I) is a DGK inhibitor (IC₅₀: 2.8 µM).

HY-N0699

Daphnoretin	Activator	99.83%
Daphnoretin (Dephnoretin), isolated from Wikstroemia indica, possesses antiviral activity.

HY-N0865

Ingenol	Activator	98.17%
Ingenol is a PKC activator, with a K_i of 30 μM, with antitumor activity.

HY-131897

1-Stearoyl-2-arachidonoyl-sn-glycerol	Activator	≥98.0%
1-Stearoyl-2-arachidonoyl-sn-glycerol is a diacylglycerol (DAG) containing polyunsaturated fatty acids.

HY-N4322

Decursinol angelate	Activator	99.54%
Decursinol angelate, a cytotoxic and protein kinase C (PKC) activating agent from the root of Angelica gigas, possesses anti-tumor and anti-inflammatory activities.

HY-108391

C8-Ceramide	Activator	≥98.0%
C8-Ceramide (N-Octanoyl-D-erythro-sphingosine) is a cell-permeable analog of naturally occurring ceramides.

HY-131648

1-Oleoyl-2-acetyl-sn-glycerol	Activator
1-Oleoyl-2-acetyl-sn glycerol is a synthetic, cell permeable diacylglycerol analog.

HY-N2180

Pinoresinol dimethyl ether	Activator	99.39%
Pinoresinol dimethyl ether ((+)-Eudesmin) is a non-phenolic furofuran lignan isolated from Magnolia biondii with neuritogenic activity.

HY-107613A

R 59-022 hydrochloride	Activator	98.88%
R 59-022 (DKGI-I) hydrochloride is a DGK inhibitor (IC₅₀: 2.8 µM).

HY-107421

Prostratin	Activator	99.32%
Prostratin, a natural terpenoid compound, is a PKC activator, with a K_i of 12.5 nM and shows inhibitory effect on HIV-1.

HY-131897S

1-Stearoyl-2-Arachidonoyl-d₈-sn-Glycerol	Activator

HY-128468

1,2-Dimyristoyl-sn-glycerol	Activator
1,2-Dimyristoyl-sn-glycerol is a saturated diacylglycerol and a weak second messenger for the activation of PKC.

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