1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. SGK
  4. SGK Inhibitors

SGK Inhibitors

SGK1

SGK3

SGK2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

SGK Inhibitors & Degraders
Product Name SGK1 SGK3 SGK2 Purity
GSK 650394
SGK1
    99.76%
EMD638683
SGK1, IC50: 3 μM
    99.94%
SGK1-IN-1
SGK1
    99.57%
PROTAC SGK3 degrader-1  
SGK3
  99.89%
SGK1-IN-9
SGK1
   
PT109
SGK1, IC50: 1.34 μM
SGK3, IC50: 26.4 μM
SGK2, IC50: 5.6 μM
99.20%
SGK1-IN-2
SGK1, IC50: 5-25 nM
    98.36%
EMD638683 (S-Form)
SGK1, IC50: > 300 nM
    99.95%
SGK1-IN-3 hydrochloride
SGK1, IC50: <1 nM
   
EMD638683 (R-Form)
SGK1
    99.86%
SGK1-IN-3
SGK1, IC50: <1 nM
   
SGK1-IN-5
SGK1, IC50: 0.003 μM
   
SGK1-IN-6
SGK1, IC50: 0.39 μM
SGK3, IC50: 1.95 μM
SGK2, IC50: 1.76 μM
PROTAC SGK3 degrader-2
SGK1, IC50: 1.4 μM
SGK3, IC50: 0.6 μM