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  2. Vitamin D Related/Nuclear Receptor
  3. Nuclear Hormone Receptor 4A/NR4A
  4. Nuclear Hormone Receptor 4A/NR4A Inhibitors

Nuclear Hormone Receptor 4A/NR4A Inhibitors

Nur77/NR4A1

Nurr1/NR4A2

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Please try each isoform separately.

Nuclear Hormone Receptor 4A/NR4A Inhibitors, Agonists, Antagonists, Activators, Modulators, Inducers & Degraders
Nombre del producto Nur77/NR4A1 Nurr1/NR4A2 Pureza
Celastrol
Nur77/NR4A1
  99.90%
Cytosporone B
Nur77/NR4A1
  99.23%
DIM-C-pPhOH
Nur77/NR4A1
  98.88%
Amodiaquine  
Nurr1/NR4A2
99.92%
Teduglutide
Nur77/NR4A1
  99.85%
DIM-3,5-Cl2
Nur77/NR4A1, Kd: 7.7 μM
Nurr1/NR4A2, Kd: 12 μM
99.18%
BI1071
Nur77/NR4A1
 
Amodiaquine dihydrochloride dihydrate  
Nurr1/NR4A2
99.92%
Amodiaquine dihydrochloride  
Nurr1/NR4A2
99.97%
TMPA
Nur77/NR4A1
  98.40%
4A7C-301  
Nurr1/NR4A2
99.86%
C-DIM12  
Nurr1/NR4A2
98.01%
NR-V04
Nur77/NR4A1
  99.90%
Glycerol kinase, microorganism
Nur77/NR4A1
 
Triptohypol C
Nur77/NR4A1
 
IP7e  
Nurr1/NR4A2
99.72%
DIM-C-pPhCO2Me
Nur77/NR4A1
  99.47%
Nurr1 agonist 2  
Nurr1/NR4A2
98.03%
Nurr1 inverse agonist-1  
Nurr1/NR4A2
98.83%
DIM-C-pPhOCH3
Nur77/NR4A1
  99.65%
Nurr1 agonist 12  
Nurr1/NR4A2, EC50: 0.06 μM
99.62%
THPN
Nur77/NR4A1
  98.00%
4-PQBH
Nur77/NR4A1
  99.14%
Nur77 modulator 1
Nur77/NR4A1
  98.61%
Nurr1 agonist 14  
Nurr1/NR4A2, EC50: 0.09 μM
99.42%
PROTAC IKKβ/NR4A1 degrader-1
Nur77/NR4A1
 
Nur77 antagonist 2
Nur77/NR4A1, Kd: 0.42 μM
 
Nur77 modulator 5
Nur77/NR4A1
 
Nur77 modulator 4
Nur77/NR4A1, Kd: 0.477 μM
 
Nur77 modulator 2
Nur77/NR4A1
 
Nur77 antagonist 1
Nur77/NR4A1
 
Nur77 modulator 6
Nur77/NR4A1
 
Nurr1 agonist 9  
Nurr1/NR4A2, EC50: 0.09 μM
Nurr1/NR4A2, Ki: 0.17 μM
Nurr1 agonist 13  
Nurr1/NR4A2, EC50: 0.06 μM
Nurr1 agonist 10  
Nurr1/NR4A2, EC50: 40 nM
Nur77 modulator 3
Nur77/NR4A1
  99.01%
Nurr1/RXR agonist 1  
Nurr1/NR4A2
Nurr1 agonist 5  
Nurr1/NR4A2
NR4A agonist-2
Nur77/NR4A1, EC50: 0.098 μM
Nurr1/NR4A2, EC50: 0.092 μM