Blue FPG-A trisodium
Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2).
For research use only. We do not sell to patients.
- CAS No.: 78617-94-4
- Formula: C29H17ClN7Na3O11S3
- Molecular Weight:840.10
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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p2x1 Receptor 35.5 μM (IC50) |
P2Y1 Receptor 2.6 μM (IC50) |
Blue FPG-A trisodium (RB 2 para) (1-100 μM) inhibits the α,β-methylene ATP (α,β-MeATP) induced contraction of the rat vas deferens (RVD) and the adenosine 5′-O-(2-thiophosphate) (ADPβS) induced relaxation of the Carbachol (HY-B1208) precontracted guinea-pig taenia coli (GPTC)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 78617-94-4
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Molecular Weight 840.10
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Formula C29H17ClN7Na3O11S3
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SMILES
O=S(C(C(N)=C1C2=O)=CC(NC3=CC=C(NC4=NC(Cl)=NC(NC5=CC=C(S(=O)(O[Na])=O)C=C5)=N4)C(S(=O)(O[Na])=O)=C3)=C1C(C6=C2C=CC=C6)=O)(O[Na])=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)