1152747-82-4
1152747-82-4
Chemical Structure
Enerisant
Synonym(s): TS-091
- CAS 番号: 1152747-82-4
- Formula:C22H30N4O3
- Molecular Weight:398.50
IUPAC Name: (R)-(1-(4-(3-(2-methylpyrrolidin-1-yl)propoxy)phenyl)-1H-pyrazol-4-yl)(morpholino)methanone
InChIKey: IABXVJILZYNSTM-GOSISDBHSA-N
SMILES: O=C(C1=CN(C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N=C1)N4CCOCC4
Biological Activity: Enerisant (TS-091) is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively[1].
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Enerisant | 99.79% | Enerisant (TS-091) is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively. | ||||||||||||||||||||
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References
Keywords
