1233248-29-7
1233248-29-7
Chemical Structure
TASP0412098
- CAS No.: 1233248-29-7
- Formula:C27H23ClN2O3
- Molecular Weight:458.94
IUPAC Name: 2-(1-(4-((4-chlorophenethyl)carbamoyl)benzyl)isoquinolin-4-yl)acetic acid
InChIKey: DAGAYHFLQZNDFS-UHFFFAOYSA-N
SMILES: O=C(CC1=CN=C(C2=C1C=CC=C2)CC3=CC=C(C=C3)C(NCCC4=CC=C(C=C4)Cl)=O)O
Biological Activity: TASP0412098 is an orally available, potent and selective CRTH2/DP2 antagonist with high binding affinity (IC50 2.1 nM) and functional activity (IC50 12 nM). TASP0412098 has the potential to suppress asthma in mouse and guinea pig bronchial asthma models[1].
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TASP0412098 | TASP0412098 is an orally available, potent and selective CRTH2/DP2 antagonist with high binding affinity (IC50 2.1 nM) and functional activity (IC50 12 nM). TASP0412098 has the potential to suppress asthma in mouse and guinea pig bronchial asthma models. | |||||||||||||||||||||
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References
Keywords
