1262032-37-0
1262032-37-0
Chemical Structure
dMeThPmR
- CAS No.: 1262032-37-0
- Formula:C12H14N2O4S
- Molecular Weight:282.32
InChIKey: MWHOUOZINAUPEL-IVZWLZJFSA-N
SMILES: O=C1N([C@H]2C[C@H](O)[C@@H](CO)O2)C=C(C=C(C)S3)C3=N1
Biological Activity: dMeThPmR, a ribonucleoside derivative, is a potent and selective human nucleoside transporter 1 (hCNT1) inhibitor (Ki = 0.3-0.98 μM). dMeThPmR exhibit weak inhibitory activity on hCNT2 (IC50 = 133 μM) and hCNT3 (Ki = 32.7 μM). dMeThPmR can protect cells from the toxicity of nucleoside drugs. dMeThPmR can be used for the research of cancer[1].
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dMeThPmR | dMeThPmR, a ribonucleoside derivative, is a potent and selective human nucleoside transporter 1 (hCNT1) inhibitor (Ki = 0.3-0.98 μM). dMeThPmR exhibit weak inhibitory activity on hCNT2 (IC50 = 133 μM) and hCNT3 (Ki = 32.7 μM). dMeThPmR can protect cells from the toxicity of nucleoside drugs. dMeThPmR can be used for the research of cancer. | |||||||||||||||||||||
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References
Keywords
