137515-05-0
Chemical Structure
RG-14467
- CAS No.: 137515-05-0
- Formula:C14H14N2O3
- Molecular Weight:258.27
IUPAC Name: 4-((2,5-dihydroxybenzyl)amino)benzamide
InChIKey: CHXLDPYIXVXZTF-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(NCC2=CC(O)=CC=C2O)C=C1)N
Biological Activity: RG-14467 is an epidermal growth factor receptor tyrosine kinase inhibitor with activity that inhibits enzyme activity. RG-14467 has similar inhibition kinetics to Lavendustin-A, with a dissociation constant of 3.4μM for the initial rapidly formed complex and an overall dissociation constant estimated to be less than or equal to 30nM, and is a partially competitive inhibitor for ATP.
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RG-14467 | RG-14467 is an epidermal growth factor receptor tyrosine kinase inhibitor with activity that inhibits enzyme activity. RG-14467 has similar inhibition kinetics to Lavendustin-A, with a dissociation constant of 3.4μM for the initial rapidly formed complex and an overall dissociation constant estimated to be less than or equal to 30nM, and is a partially competitive inhibitor for ATP. | |||||||||||||||||||||
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Keywords
