143257-98-1
143257-98-1
Chemical Structure
Lerisetron
- CAS No.: 143257-98-1
- Formula:C18H20N4
- Molecular Weight:292.38
IUPAC Name: 1-benzyl-2-(piperazin-1-yl)-1H-benzo[d]imidazole
InChIKey: PWWDCRQZITYKDV-UHFFFAOYSA-N
SMILES: C1(N=C(N2CCNCC2)N3CC4=CC=CC=C4)=C3C=CC=C1
Biological Activity: Lerisetron is a potent 5-HT3 antagonists and possess high-affinity binding for the 5-HT3 receptors with pKi value of 9.2. Lerisetron has a potent ability to inhibit the 5-HT-evoked reflex bradycardia in urethane-anesthetized rats[1].
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Lerisetron | 99.69% | Lerisetron is a potent 5-HT3 antagonists and possess high-affinity binding for the 5-HT3 receptors with pKi value of 9.2. Lerisetron has a potent ability to inhibit the 5-HT-evoked reflex bradycardia in urethane-anesthetized rats. | ||||||||||||||||||||
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Lerisetron (Standard) | ≥98% | Lerisetron (Standard) is the analytical standard of Lerisetron. This product is intended for research and analytical applications. Lerisetron is a potent 5-HT3 antagonists and possess high-affinity binding for the 5-HT3 receptors with pKi value of 9.2. Lerisetron has a potent ability to inhibit the 5-HT-evoked reflex bradycardia in urethane-anesthetized rats. | ||||||||||||||||||||
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References
Keywords
