1478364-87-2
1478364-87-2
Chemical Structure
PXS-4681A
- CAS No.: 1478364-87-2
- Formula:C10H14ClFN2O3S
- Molecular Weight:296.75
IUPAC Name: (Z)-4-((2-(aminomethyl)-3-fluoroallyl)oxy)benzenesulfonamide hydrochloride
InChIKey: VBGNJMUEMDYZJJ-HGKIGUAWSA-N
SMILES: O=S(C1=CC=C(OC/C(CN)=C\F)C=C1)(N)=O.Cl
Biological Activity: PXS-4681A is a potent, selective, irreversible and orally active semicarbazide-sensitive amine oxidase (SSAO; VAP-1) inhibitor with a Ki of 37 nM. PXS-4681A shows highly selectivity over related amine oxidases, ion channels, and seven-transmembrane domain receptors. PXS-4681A has anti-inflammatory effects[1].
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PXS-4681A | 99.40% | PXS-4681A is a potent, selective, irreversible and orally active semicarbazide-sensitive amine oxidase (SSAO; VAP-1) inhibitor with a Ki of 37 nM. PXS-4681A shows highly selectivity over related amine oxidases, ion channels, and seven-transmembrane domain receptors. PXS-4681A has anti-inflammatory effects. | ||||||||||||||||||||
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References
Keywords
