155649-00-6
Chemical Structure
PG 9 maleate
- CAS No.: 155649-00-6
- Formula:C21H26BrNO6
- Molecular Weight:468.34
IUPAC Name: (1R,3r,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl 2-(4-bromophenyl)propanoate maleate
InChIKey: VBUSCULTLLOSLM-QFWARMDFSA-N
SMILES: O=C(C(C1=CC=C(Br)C=C1)C)O[C@H]2C[C@H]3CC[C@H](N3C)C2.O=C(O)/C=C\C(O)=O
Biological Activity: PG 9 maleate is a compound with analgesic and anti-memory loss activity. PG 9 maleate exerts analgesic effects by enhancing central cholinergic transmission. PG 9 maleate protects against memory loss caused by scopolamine or dicyclomine within a specific dose range. The affinity profile of PG 9 maleate indicates significant selectivity among the M4/M1 receptor subtypes, which may be the mechanism for its analgesic and anti-memory loss effects. PG 9 maleate can increase the release of acetylcholine, thereby improving its biological activity[1].
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PG 9 maleate | PG 9 maleate is a compound with analgesic and anti-memory loss activity. PG 9 maleate exerts analgesic effects by enhancing central cholinergic transmission. PG 9 maleate protects against memory loss caused by scopolamine or dicyclomine within a specific dose range. The affinity profile of PG 9 maleate indicates significant selectivity among the M4/M1 receptor subtypes, which may be the mechanism for its analgesic and anti-memory loss effects. PG 9 maleate can increase the release of acetylcholine, thereby improving its biological activity. | |||||||||||||||||||||
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Keywords
