1669444-50-1
1669444-50-1
Chemical Structure
PF-05214030
- CAS No.: 1669444-50-1
- Formula:C17H13Cl2FN2O4S
- Molecular Weight:431.27
InChIKey: RZAIRBXIVAVGHE-UHFFFAOYSA-N
SMILES: N#CC1=CC=C(C=C1F)OCC2(CN(S(=O)(C3=CC=C(C=C3Cl)Cl)=O)C2)O
Biological Activity: PF-05214030 is a TRPV4 antagonist (IC50: 4 and 27nM for hTRPV4 and rTRPV4 respectively). PF-05214030 reverses the reduction in bladder capacity caused by intravesical infusion of a TRPV4 agonist[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PF-05214030 | 99.81% | PF-05214030 is a TRPV4 antagonist (IC50: 4 and 27nM for hTRPV4 and rTRPV4 respectively). PF-05214030 reverses the reduction in bladder capacity caused by intravesical infusion of a TRPV4 agonist. | ||||||||||||||||||||
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References
Keywords
