1808389-92-5
1808389-92-5
Chemical Structure
GABAA receptor agent 5
- CAS No.: 1808389-92-5
- Formula:C21H25N3O2S
- Molecular Weight:383.51
IUPAC Name: N-(3-(3,9-diazaspiro[5.5]undecane-3-carbonyl)phenyl)thiophene-2-carboxamide
InChIKey: PQGDUNWRHHLMNT-UHFFFAOYSA-N
SMILES: O=C(C1=CC=CS1)NC2=CC=CC(C(N3CCC4(CC3)CCNCC4)=O)=C2
Biological Activity: GABAA receptor agent 5 (compound 018) is a potent γ-GABAAR antagonist with an Ki of 0.020 µM. GABAA receptor agent 5 shows γ-GABAAR antagonist activity with low cellular membrane permeability[1].
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GABAA receptor agent 5 | GABAA receptor agent 5 (compound 018) is a potent γ-GABAAR antagonist with an Ki of 0.020 µM. GABAA receptor agent 5 shows γ-GABAAR antagonist activity with low cellular membrane permeability. | |||||||||||||||||||||
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References
Keywords
