1839519-57-1
1839519-57-1
Chemical Structure
Br-PBTC
- CAS No.: 1839519-57-1
- Formula:C14H15BrN2OS
- Molecular Weight:339.25
IUPAC Name: (R)-7-bromo-N-(piperidin-3-yl)benzo[b]thiophene-2-carboxamide
InChIKey: LRYYPTVUWGMZQB-SNVBAGLBSA-N
SMILES: O=C(C1=CC2=CC=CC(Br)=C2S1)N[C@H]3CNCCC3
Biological Activity: Br-PBTC is a potent, 2/4 subtype-selective positive allosteric modulator of nAChRs (nicotinic acetylcholine receptors) with α2β2, α2β4, α4β2, α4β4, (α4β2)2α4 and (α4β2)2β2 EC50 ranges from 0.1-0.6 μM. Br-PBTC acts from the c-tail of an α subunit[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Br-PBTC | 98.0% | Br-PBTC is a potent, 2/4 subtype-selective positive allosteric modulator of nAChRs (nicotinic acetylcholine receptors) with α2β2, α2β4, α4β2, α4β4, (α4β2)2α4 and (α4β2)2β2 EC50 ranges from 0.1-0.6 μM. Br-PBTC acts from the c-tail of an α subunit. | ||||||||||||||||||||
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References
Keywords
